Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HMFFXQOXUNOHJJ
|
9.4 | IC50 | 2 | — | |
RVQPBMWIXPQVNW
|
9.4 | Ki | 3 | — | |
ABHCOFKCKYHXPW
|
9.3 | IC50 | 2 | — | |
QIOKOIIOOCXZFW
|
9.3 | IC50 | 3 | — | |
GXSHWBSAHCQKFV
|
9.3 | IC50 | 3 | — | |
VBVOCYOFXNIYLW
|
9.3 | IC50 | 2 | — | |
ZGTXKDRQZHGJAA
|
9.3 | Ki | 3 | — | |
PKSWBZKUKRFMGK
|
9.3 | IC50 | 2 | — | |
GAMSTIVHSDPIFY
|
9.3 | Ki | 3 | — | |
MWNNSAODMZRACW
|
9.3 | Ki | 3 | — | |
RVBJJKHDYYRLRK
|
9.3 | Ki | 3 | — | |
NUQNGPSYNHDQBA
|
9.3 | Ki | 3 | — | |
AKSPXUYBVOVPHA
|
9.3 | IC50 | 2 | — | |
AUSOZFFBBXRILI
|
9.3 | Ki | 3 | — | |
BQVZFNYKORVNKX
|
9.3 | Ki | 3 | — | |
GFWDUDFEFKZZQI
|
9.3 | Ki | 3 | — | |
NIRPQZMBABINPZ
|
9.3 | Ki | 3 | — | |
NQXPYPBIBFFEAE
|
9.3 | IC50 | 2 | — | |
PXZVRKSGUYKVGK
|
9.3 | IC50 | 2 | — | |
TUMIEGHWQWSXPG
|
9.3 | IC50 | 3 | — | |
UOMPPOVQMYNXST
|
9.3 | IC50 | 2 | — | |
WRMDZFXPBIHCOL
|
9.3 | IC50 | 2 | — | |
CALQCAQZMQRBIJ
|
9.3 | Ki | 3 | — | |
JKCKHRWRMSOFHW
|
9.3 | IC50 | 2 | — | |
OVTVOGQQMFPUDP
|
9.3 | Ki | 3 | — | |
RFEQCBHECCTMEH
|
9.3 | Ki | 3 | — | |
XXPYNUSOQUYFNM
|
9.3 | IC50 | 2 | — | |
IYFHLODASXJRCX
|
9.3 | Ki | 3 | — | |
XERUWQHYFFRDQN
|
9.3 | IC50 | 3 | — | |
BZUBDLKATGBRRF
|
9.3 | IC50 | 2 | — | |
DEQPQIXEUNLWAL
|
9.3 | IC50 | 2 | — | |
HLPARXMUJBJYFM
|
9.3 | IC50 | 2 | — | |
NIPDJBAMYWKEHF
|
9.3 | IC50 | 2 | — | |
DEJOUBIDXHXKJV
|
9.2 | IC50 | 2 | — | |
JUDXZPPDZZPKEK
|
9.2 | IC50 | 3 | — | |
NEBCCMOWOJKFFS
|
9.2 | IC50 | 3 | — | |
OZWQMYWGAMLKRZ
|
9.2 | IC50 | 2 | — | |
FTLPJRYZRTWCHZ
|
9.2 | Ki | 3 | — | |
KDBWXGCLBVMYIK
|
9.2 | IC50 | 3 | — | |
YVBZACMJRRMNCT
|
9.2 | Ki | 3 | — | |
SDHRADPEFDLIKD
|
9.2 | IC50 | 3 | — | |
DDQXBYGNFGPJRL
|
9.2 | IC50 | 3 | — | |
FAUDAQJUMHDILO
|
9.2 | IC50 | 2 | — | |
OKUXRVPIXCSROX
|
9.2 | Ki | 2 | — | |
RDRLFKLJQDCWPH
|
9.2 | IC50 | 2 | — | |
RMGUESBYRVXIQU
|
9.2 | IC50 | 2 | — | |
XVTCHURPFKMJKZ
|
9.2 | IC50 | 2 | — | |
YJMUKULIAJBLOM
|
9.2 | Ki | 3 | — | |
ZJFKGQNBMRSSPS
|
9.2 | Ki | 3 | — | |
HXUHHDBYIBYXPB
|
9.2 | IC50 | 3 | — |