Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KMIKZMJCDRKNJE
|
11.7 | Ki | 3 | — | |
RJBLYAOGZIACGS
|
11.7 | Ki | 3 | — | |
BEXSRDRFSVXXPU
|
11.5 | Ki | 3 | — | |
GZHPOGVPEBAKBW
|
11.3 | Ki | 3 | — | |
GAPPKQMJLOBLDJ
|
11.2 | IC50 | 3 | — | |
TWIFKBILIHXMMI
|
11.2 | Ki | 3 | — | |
UCLIZEJSCGLLJP
|
11.2 | Ki | 3 | — | |
XCEBXSIYXWIQPP
|
11.2 | Ki | 3 | — | |
FLWOSIOISGGQGY
|
11.1 | Ki | 2 | — | |
VKNMCBUJJJKJQM
|
11.1 | Ki | 3 | — | |
AUYCDANENPJVBH
|
11.0 | IC50 | 3 | — | |
DXFVPMMMQNXSOZ
|
11.0 | Ki | 3 | — | |
JIRRCQJZLNTIIP
|
11.0 | IC50 | 3 | — | |
LLNGTXPGUYSOTJ
|
11.0 | IC50 | 3 | — | |
RCZYLHFODBPYHX
|
11.0 | IC50 | 3 | — | |
UEYVMWQIHAGSEU
|
11.0 | IC50 | 3 | — | |
VHHMNEWIYJHDIY
|
11.0 | Ki | 3 | — | |
CDQXYOYHHLAARJ
|
11.0 | Ki | 3 | — | |
OGLBDVCMFBBNFL
|
10.9 | Ki | 3 | — | |
DVKOJQHRIKGCMQ
|
10.9 | IC50 | 2 | — | |
XWOSSDMMJDYDBX
|
10.9 | Ki | 3 | — | |
OYVCFKLZLLYNOW
|
10.8 | Ki | 3 | — | |
BAUZKJYZGGFFLL
|
10.8 | Ki | 3 | — | |
ZNOTUHKIYPIPHI
|
10.8 | Ki | 3 | — | |
PRDCOFAMJJLIRA
|
10.8 | Ki | 3 | — | |
APJNEWHEOPKPSA
|
10.7 | Ki | 3 | — | |
ADHFWXANXDIZPQ
|
10.7 | Ki | 3 | — | |
BLHWEGXFMWEIHN
|
10.7 | IC50 | 3 | — | |
BUSRDZKIQOWUOO
|
10.7 | IC50 | 3 | — | |
FKRJLOFLENGVAA
|
10.7 | IC50 | 3 | — | |
FKRJLOFLENGVAA
|
10.7 | IC50 | 3 | — | |
FVOUGHZKLGXVGD
|
10.7 | IC50 | 3 | — | |
GGOYZNQGGMFQKZ
|
10.7 | IC50 | 3 | — | |
GRHJHFJDNAZVLO
|
10.7 | IC50 | 3 | — | |
HTPLJVYJVSGLKR
|
10.7 | IC50 | 3 | — | |
ITPBXRZSRGMCKW
|
10.7 | IC50 | 3 | — | |
JEVIKKKBDOXJFA
|
10.7 | Ki | 3 | — | |
KEQAECANTREWKS
|
10.7 | IC50 | 3 | — | |
KNZWOEPEIQKBJT
|
10.7 | IC50 | 3 | — | |
LDKXEQFXIGEBKS
|
10.7 | IC50 | 3 | — | |
LGIGKYXJCHINMH
|
10.7 | IC50 | 3 | — | |
LKVRXZVHFRHSKB
|
10.7 | IC50 | 3 | — | |
LQSXQOIVFCNKGT
|
10.7 | IC50 | 3 | — | |
LWXCNBLYXPLROO
|
10.7 | IC50 | 3 | — | |
MCHAJIZUZNPBCS
|
10.7 | Ki | 3 | — | |
MDSSZYNUYNBVFZ
|
10.7 | IC50 | 2 | — | |
MMQGQQIWWVVFQW
|
10.7 | IC50 | 3 | — | |
MRSQWVHHJSPXOI
|
10.7 | IC50 | 3 | — | |
PAKQZSJYQOIVOH
|
10.7 | Ki | 3 | — | |
RZULTVPKWRBATD
|
10.7 | IC50 | 3 | — |