Target Details
| UniProt AC | P11274 |
|---|---|
| Gene Symbol | BCR |
| Protein Name | Breakpoint cluster region protein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF09036 (Bcr-Abl_Oligo) PF00168 (C2) PF19057 (PH_19) PF00620 (RhoGAP) PF00621 (RhoGEF) |
Summary
- Multi-target molecules 338
- Clinical molecules 25
- Avg pChEMBL 7.32
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (338)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NOASFNUCHAXHFR
|
6.2 | IC50 | 2 | — | |
GHOABOFWXUXZRJ
|
6.2 | IC50 | 2 | — | |
VTLBOGLRMDPIDX
|
6.2 | IC50 | 2 | — | |
XTAVRPBOWLIGCW
|
6.2 | IC50 | 2 | — | |
CCAIGJJHLPYVQD
|
6.2 | IC50 | 2 | — | |
RSMXWAAHBXSACS
|
6.2 | IC50 | 2 | — | |
HDTCSYZQKDPDHW
|
6.2 | IC50 | 3 | — | |
SPUAKYCGPJOVBW
|
6.2 | IC50 | 2 | — | |
LNMRSSIMGCDUTP
|
6.2 | Kd | 13 | — | |
XPWDRROAEFMYOQ
|
6.2 | IC50 | 2 | — | |
OMZCMEYTWSXEPZ
|
6.2 | Kd | 43 | Yes | |
UQRCJCNVNUFYDX
|
6.2 | Kd | 27 | — | |
ZQTRXPRIWRFHRY
|
6.2 | IC50 | 2 | — | |
YCCAMNPZGLARRQ
|
6.1 | IC50 | 2 | — | |
FNHKPVJBJVTLMP
|
6.1 | Kd | 29 | — | |
SPBYVRXRBROCFD
|
6.1 | IC50 | 2 | — | |
FQRASLPAVXFUEP
|
6.1 | IC50 | 2 | — | |
RBVZQGGIPAKNKY
|
6.1 | IC50 | 2 | — | |
JLNFEMZJZFVZHH
|
6.1 | IC50 | 2 | — | |
YVLLRTOXLOIJHL
|
6.1 | IC50 | 2 | — | |
ULUNCQWGUQFHNV
|
6.1 | IC50 | 4 | — | |
YVNKPHLJKPWZRT
|
6.1 | IC50 | 4 | — | |
PIGRLCPKGBFTPO
|
6.1 | IC50 | 2 | — | |
YRCHYHRCBXNYNU
|
6.1 | Kd | 13 | — | |
DTMQLWYGSUIGTJ
|
6.1 | IC50 | 2 | — | |
UHTHHESEBZOYNR
|
6.1 | Kd | 66 | Yes | |
YZNIHXUBUWEUCM
|
6.1 | IC50 | 14 | — | |
ZJWPYYIRORJZPQ
|
6.1 | IC50 | 4 | — | |
JMCVXZQETOMXJG
|
6.0 | IC50 | 2 | — | |
BCUJRVQSIFNOKH
|
6.0 | IC50 | 2 | — | |
CNUQKCFZQUWMFJ
|
6.0 | IC50 | 2 | — | |
OFBWCZMTFNTSHE
|
6.0 | IC50 | 3 | — | |
LIMBOIOWYJOOIC
|
6.0 | IC50 | 3 | Yes | |
QGIRAHZKAGRURU
|
6.0 | IC50 | 4 | — | |
ROFRUHKNTPJICR
|
6.0 | IC50 | 2 | — | |
RUDJLSWOUHMLOU
|
6.0 | IC50 | 3 | — | |
SPYAHPCGCDDALM
|
6.0 | IC50 | 2 | — | |
YCDIUFZXJOHIGE
|
6.0 | IC50 | 2 | — |