Target Details
| UniProt AC | P11274 |
|---|---|
| Gene Symbol | BCR |
| Protein Name | Breakpoint cluster region protein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF09036 (Bcr-Abl_Oligo) PF00168 (C2) PF19057 (PH_19) PF00620 (RhoGAP) PF00621 (RhoGEF) |
Summary
- Multi-target molecules 338
- Clinical molecules 25
- Avg pChEMBL 7.32
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (338)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CDRNAUYQMWZXOE
|
6.5 | IC50 | 2 | — | |
BFXBZGCCVBJKPX
|
6.5 | IC50 | 2 | — | |
OGRGVSAACLPSGE
|
6.5 | IC50 | 2 | — | |
ONIQOQHATWINJY
|
6.5 | Kd | 25 | — | |
FOIYVDLETGQHDE
|
6.5 | IC50 | 2 | — | |
HNAIZJDQDDXEGC
|
6.5 | IC50 | 6 | Yes | |
DDLPXZXBWGJRGK
|
6.5 | IC50 | 4 | — | |
WKBRCCPYCFUNGN
|
6.4 | IC50 | 2 | — | |
HCZZACRTGWSLPL
|
6.4 | IC50 | 6 | Yes | |
CWILIZPMLKHDKP
|
6.4 | IC50 | 2 | — | |
OGWDTZBATVFCOT
|
6.4 | IC50 | 2 | — | |
RVMLNNCKNCFOFH
|
6.4 | IC50 | 4 | — | |
SNVFOGVFJDTZIR
|
6.4 | IC50 | 2 | — | |
WVXNSAVVKYZVOE
|
6.4 | Kd | 92 | — | |
FKCRUIWBTDNJFG
|
6.4 | IC50 | 4 | — | |
MLAIONZVQZBMNT
|
6.4 | Kd | 3 | — | |
IHMRQAKZJBZCIN
|
6.4 | IC50 | 2 | — | |
UOEJSOXEHKCNAE
|
6.4 | IC50 | 4 | — | |
ZVXCXEJBPDCMRL
|
6.4 | IC50 | 3 | Yes | |
MWKSRKSEWLRPBL
|
6.4 | Kd | 1075 | — | |
DRNRCLNUHIQXOJ
|
6.4 | IC50 | 4 | — | |
ULMWPPWTYJYKFS
|
6.4 | IC50 | 2 | — | |
BCQMLQGCVHMBRI
|
6.4 | IC50 | 3 | — | |
RIWKVLUOTMXONS
|
6.4 | IC50 | 5 | — | |
ZYJKIIOWFQYSQR
|
6.4 | IC50 | 2 | — | |
VXPRMSHSUFWMNM
|
6.3 | IC50 | 2 | — | |
YDUUIKKCZDDRLN
|
6.3 | IC50 | 4 | — | |
IRABBTBTKJUYTE
|
6.3 | IC50 | 2 | — | |
BZSOOFCPERGONN
|
6.3 | IC50 | 2 | — | |
XTWQOJKEOSZUSS
|
6.3 | IC50 | 2 | — | |
AATUFOXFWPLFGG
|
6.3 | IC50 | 2 | — | |
MZJIJJIHVGGOAC
|
6.3 | IC50 | 3 | Yes | |
NJIYAJRNLNJIGY
|
6.3 | IC50 | 2 | — | |
OONFNUWBHFSNBT
|
6.3 | Kd | 11 | — | |
PMXPPBGETIGOHR
|
6.3 | IC50 | 2 | — | |
BQQYXPHRXIZMDM
|
6.3 | IC50 | 3 | — | |
DHQCZYDRYAFSAN
|
6.3 | IC50 | 2 | — | |
HFBBNWGIUOYGEZ
|
6.3 | Kd | 2 | — | |
NUMDANVMMRMHHS
|
6.3 | IC50 | 2 | — | |
KTUFNOKKBVMGRW
|
6.3 | IC50 | 3 | — | |
PGNPRFGVXQKJFG
|
6.3 | IC50 | 4 | — | |
TWPHWLKUNGVMCP
|
6.2 | IC50 | 2 | — | |
ZLPLPSSLKIOLRR
|
6.2 | IC50 | 2 | — | |
GYTPDENASJFHSZ
|
6.2 | IC50 | 2 | — | |
ODPGGGTTYSGTGO
|
6.2 | IC50 | 153 | — | |
UKTICNMOUVEYRR
|
6.2 | IC50 | 4 | — | |
UXRUDXZNSIAVNZ
|
6.2 | IC50 | 2 | — | |
LCQYMDMUCJFFKN
|
6.2 | IC50 | 5 | Yes | |
LYPYSTQHYJMALD
|
6.2 | Kd | 2 | — | |
MDYKWTJHVLZUAH
|
6.2 | IC50 | 2 | — |