Target Details
| UniProt AC | P11274 |
|---|---|
| Gene Symbol | BCR |
| Protein Name | Breakpoint cluster region protein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF09036 (Bcr-Abl_Oligo) PF00168 (C2) PF19057 (PH_19) PF00620 (RhoGAP) PF00621 (RhoGEF) |
Summary
- Multi-target molecules 338
- Clinical molecules 25
- Avg pChEMBL 7.32
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (338)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WTKZJFUSCLBZBH
|
6.9 | IC50 | 2 | — | |
WKDACQVEJIVHMZ
|
6.9 | Kd | 46 | — | |
DMELXOVEWUBBNG
|
6.8 | IC50 | 2 | — | |
GPBIUFSBAGPHFC
|
6.8 | IC50 | 2 | — | |
ULSOOODMFMCIIK
|
6.8 | IC50 | 2 | — | |
FXYAYKHUOYATRN
|
6.8 | IC50 | 2 | — | |
MKVWYGFIMREUPS
|
6.8 | IC50 | 2 | — | |
PMKFHRVILXSTGE
|
6.8 | IC50 | 2 | — | |
QOFWWNRCEIPMLU
|
6.8 | IC50 | 4 | Yes | |
LOLPPWBBNUVNQZ
|
6.8 | Kd | 97 | Yes | |
SPMVMDHWKHCIDT
|
6.8 | Kd | 30 | — | |
DQXHCIXMRVKNKN
|
6.8 | IC50 | 2 | — | |
JXSFGZPUWDXKPG
|
6.8 | IC50 | 2 | — | |
JMHFJMQAYNDVED
|
6.8 | IC50 | 2 | — | |
KTUFNOKKBVMGRW
|
6.8 | IC50 | 38 | Yes | |
YYBHKLYUXAWHPX
|
6.8 | IC50 | 2 | — | |
RITAVMQDGBJQJZ
|
6.7 | Kd | 43 | — | |
SCLMNCGKQRDXNW
|
6.7 | IC50 | 2 | — | |
GJNWPXMEFQRJIZ
|
6.7 | IC50 | 2 | — | |
DXELIKRBLYYPBN
|
6.7 | IC50 | 2 | — | |
JAGCFIAIQQJIFB
|
6.7 | IC50 | 2 | — | |
JYSOTWILHTUWTB
|
6.7 | IC50 | 2 | — | |
MBAORQXUHJBLIE
|
6.7 | IC50 | 2 | — | |
OOTFJNZUPSBENC
|
6.7 | IC50 | 2 | — | |
PFBROONURYHZHV
|
6.7 | IC50 | 2 | — | |
SZJRFGYYRZITCZ
|
6.7 | IC50 | 4 | — | |
UDHQGXCXSRGAPA
|
6.7 | IC50 | 4 | — | |
FCCJIRJUDAWXRO
|
6.7 | IC50 | 4 | — | |
JMMFXXPAQAEXJE
|
6.7 | IC50 | 2 | — | |
OKFQCGQMFZAGPH
|
6.7 | IC50 | 2 | — | |
DSTHNGDWKODQRN
|
6.7 | IC50 | 2 | — | |
HVFUJLVTNVRIEV
|
6.7 | IC50 | 2 | — | |
MAEVHSVRMUAWLW
|
6.7 | IC50 | 2 | — | |
ZCCPLJOKGAACRT
|
6.6 | Kd | 599 | — | |
KYENXKDRIQKRJP
|
6.6 | IC50 | 5 | — | |
BNQMUNINUMWZQI
|
6.6 | IC50 | 2 | — | |
FDKRVDGCRVDZMG
|
6.6 | IC50 | 2 | — | |
ITBOQKWIUSIIGU
|
6.6 | IC50 | 2 | — | |
WEVYNIUIFUYDGI
|
6.6 | IC50 | 2 | — | |
BYQSNNVPDUUJAX
|
6.6 | IC50 | 2 | — | |
UDAPJMBKYNTXRB
|
6.6 | IC50 | 2 | — | |
VUYWDRJRXVAGSK
|
6.6 | IC50 | 3 | — | |
MRCMFAWPPPUHNS
|
6.5 | IC50 | 2 | — | |
ZJOODAFPLSLHSN
|
6.5 | IC50 | 2 | — | |
DIZCOWFZHJWMBP
|
6.5 | IC50 | 2 | — | |
VWMJHAFYPMOMGF
|
6.5 | Kd | 15 | — | |
QJYIYSNZNFDPHG
|
6.5 | IC50 | 2 | — | |
SPWAAJJVMPKJIU
|
6.5 | IC50 | 2 | — | |
XZXHXSATPCNXJR
|
6.5 | Kd | 165 | Yes | |
BSVDGQDTPDLQCS
|
6.5 | IC50 | 2 | — |