Target Details
| UniProt AC | P11274 |
|---|---|
| Gene Symbol | BCR |
| Protein Name | Breakpoint cluster region protein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF09036 (Bcr-Abl_Oligo) PF00168 (C2) PF19057 (PH_19) PF00620 (RhoGAP) PF00621 (RhoGEF) |
Summary
- Multi-target molecules 338
- Clinical molecules 25
- Avg pChEMBL 7.32
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (338)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HFGUPJNHEPCEHX
|
7.3 | IC50 | 3 | — | |
QOHRZEWGDUREJV
|
7.3 | IC50 | 2 | — | |
TWCOARREJINKIL
|
7.3 | IC50 | 2 | — | |
WVFIZRNACLGJDI
|
7.3 | IC50 | 2 | — | |
TYVQJCSBHJOJCN
|
7.3 | IC50 | 2 | — | |
QEWJRTUCCOIWLO
|
7.2 | IC50 | 2 | — | |
BLYRPGBSIKAIAU
|
7.2 | IC50 | 24 | Yes | |
HWZFQQYDALNGQT
|
7.2 | Kd | 3 | — | |
OHHSWQIUXWNAGL
|
7.2 | IC50 | 2 | — | |
RJEOZKIUSOFSDC
|
7.2 | IC50 | 2 | — | |
SYMMGQMCJOZALT
|
7.2 | IC50 | 2 | — | |
BLOQVLVYNHGRHT
|
7.2 | IC50 | 2 | — | |
QOSZUVFISSPGCO
|
7.2 | IC50 | 2 | — | |
YZLKFFPFWYDBEB
|
7.2 | IC50 | 3 | — | |
BMCKWRUTJXVUFF
|
7.2 | IC50 | 4 | — | |
JMGXJHWTVBGOKG
|
7.2 | Kd | 7 | — | |
BFDYMLHRCBEGCZ
|
7.2 | IC50 | 2 | — | |
IORXBTIJLGQAEJ
|
7.2 | IC50 | 2 | — | |
USMCKQQKWYXXCV
|
7.2 | IC50 | 2 | — | |
ZFTWKPRQHPMJAA
|
7.2 | IC50 | 2 | — | |
BFSMWDPRHAHFSS
|
7.1 | IC50 | 2 | — | |
IDMLCHSTWFWJHX
|
7.1 | IC50 | 2 | — | |
DDRLQMSTWJRCMI
|
7.1 | IC50 | 2 | — | |
WJEOLQLKVOPQFV
|
7.1 | Kd | 24 | — | |
KFUPFXKVTHKTDP
|
7.1 | IC50 | 2 | — | |
PSKGMHXAYOCLLX
|
7.1 | IC50 | 2 | — | |
GKLDJIUKRHJMHG
|
7.1 | IC50 | 2 | — | |
AZCFXTPLBWULJY
|
7.1 | IC50 | 2 | — | |
ZAXFYYCHCGZIPG
|
7.1 | IC50 | 2 | — | |
FZXLZZAXHCHSEG
|
7.1 | IC50 | 2 | — | |
IAYGCINLNONXHY
|
7.1 | Kd | 50 | — | |
KEQJVXCNVVFRCN
|
7.1 | IC50 | 2 | — | |
JONUUBFCZUAOFY
|
7.0 | IC50 | 10 | — | |
NQRWHNMIXKRPES
|
7.0 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
7.0 | IC50 | 408 | — | |
HUNGUWOZPQBXGX
|
7.0 | IC50 | 4 | — | |
JHMBUEWQJDGKGS
|
7.0 | IC50 | 7 | Yes | |
OIMJFVHFGBCRHO
|
7.0 | IC50 | 2 | — | |
SWXHXBQROFJLND
|
7.0 | IC50 | 2 | — | |
CXQHYVUVSFXTMY
|
7.0 | Kd | 154 | — | |
JFLHOEAKUBGSFZ
|
7.0 | IC50 | 2 | — | |
LEPJLENCQXRNFB
|
7.0 | IC50 | 2 | — | |
VITWTRRNFRBXSR
|
7.0 | IC50 | 2 | — | |
BJBTYWHXCARYTA
|
7.0 | IC50 | 2 | — | |
HVXKQKFEHMGHSL
|
7.0 | Kd | 21 | — | |
HBROJOMCQONOAW
|
6.9 | IC50 | 2 | — | |
IQTSERMRWSERDI
|
6.9 | Kd | 3 | — | |
ASJUWXZPJDVCQZ
|
6.9 | IC50 | 2 | — | |
DDQYAVSQXTUITB
|
6.9 | IC50 | 2 | — | |
WRHJJVUSHYOUBB
|
6.9 | IC50 | 2 | — |