Target Details
| UniProt AC | P11274 |
|---|---|
| Gene Symbol | BCR |
| Protein Name | Breakpoint cluster region protein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF09036 (Bcr-Abl_Oligo) PF00168 (C2) PF19057 (PH_19) PF00620 (RhoGAP) PF00621 (RhoGEF) |
Summary
- Multi-target molecules 338
- Clinical molecules 25
- Avg pChEMBL 7.32
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (338)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CDXRBIMKCWWDMY
|
7.8 | IC50 | 2 | — | |
CJZDHNAPSGIJPC
|
7.8 | IC50 | 2 | — | |
FOYDGOBFRZQHEU
|
7.8 | IC50 | 13 | — | |
NVRXTLZYXZNATH
|
7.8 | IC50 | 47 | Yes | |
VWCSBXLDSKERLY
|
7.7 | IC50 | 2 | — | |
LHVHGXVPJPMLFB
|
7.7 | IC50 | 2 | — | |
JRJBXDYPYRFVHH
|
7.7 | IC50 | 2 | — | |
KODAMADJHOKWQH
|
7.7 | IC50 | 2 | — | |
QMWCOMCAODPOMZ
|
7.7 | IC50 | 2 | — | |
UPZUOJCELONEIR
|
7.7 | IC50 | 2 | — | |
QPEWSVDGDKWHMX
|
7.7 | IC50 | 2 | — | |
YJQOQJNKFYBZOV
|
7.7 | IC50 | 2 | — | |
YKDNQUNPTIJKCH
|
7.7 | IC50 | 2 | — | |
CBMGZXHASOIHSW
|
7.7 | IC50 | 2 | — | |
SWYGYHUKYVHTHP
|
7.7 | IC50 | 2 | — | |
YZMSPABNYFHEHD
|
7.7 | IC50 | 2 | — | |
BMFUIUDLVMJYGT
|
7.7 | IC50 | 3 | — | |
JXYHYYBXKLTNGG
|
7.7 | IC50 | 3 | — | |
AZTXEXSCWBYKOB
|
7.7 | IC50 | 2 | — | |
MIARGORLLRWINC
|
7.7 | IC50 | 2 | — | |
JBPBNXCKEHXPOS
|
7.6 | IC50 | 2 | — | |
MLSMCXWBTQUJBM
|
7.6 | IC50 | 2 | — | |
IQIXKGNNKIOWHL
|
7.6 | IC50 | 2 | — | |
OMVOXDNRIIIPHG
|
7.6 | IC50 | 2 | — | |
XESOUPPNAWVWAG
|
7.6 | IC50 | 2 | — | |
RVVOZOVEPBDKNY
|
7.6 | IC50 | 2 | — | |
GUEFRZZGCQAGLR
|
7.5 | IC50 | 2 | — | |
JLQPVUJUCFSACM
|
7.5 | IC50 | 2 | — | |
QFKVEVOGGCTCKS
|
7.5 | IC50 | 2 | — | |
OKHCJZLKVVFPLZ
|
7.5 | IC50 | 2 | — | |
JKZZCHSVFXZBAI
|
7.5 | IC50 | 6 | — | |
RIXBMLAVFFOVIP
|
7.5 | IC50 | 2 | — | |
DZFZXPPHBWCXPQ
|
7.5 | Kd | 12 | — | |
JJFYUQKAJYRNHL
|
7.5 | IC50 | 2 | — | |
NMMIVVLEPHGUEV
|
7.5 | IC50 | 2 | — | |
XKFTZKGMDDZMJI
|
7.5 | IC50 | 8 | Yes | |
QDXRELOFIZDHGS
|
7.4 | IC50 | 2 | — | |
HHZIURLSWUIHRB
|
7.4 | IC50 | 57 | Yes | |
XPWYQHDVNYIXSF
|
7.4 | IC50 | 2 | — | |
DKNUPRMJNUQNHR
|
7.4 | Kd | 33 | — | |
XLMBXWNZLPFUQW
|
7.4 | IC50 | 2 | — | |
PPMFZQWMHKWFPZ
|
7.4 | IC50 | 2 | — | |
JIBBGYSUSKAPDY
|
7.4 | IC50 | 19 | — | |
YQXVNNKJNHKVLW
|
7.4 | Kd | 3 | — | |
XEXBRZPNVDDJRA
|
7.4 | IC50 | 2 | — | |
YTOXAXYCYYWBRD
|
7.4 | IC50 | 2 | — | |
ONYASORTFKFDEA
|
7.3 | IC50 | 2 | — | |
GCIKSSRWRFVXBI
|
7.3 | Ki | 109 | Yes | |
UKHOXYCPBAGGAN
|
7.3 | Kd | 3 | — | |
VPZGFKSLFAEGRG
|
7.3 | IC50 | 2 | — |