Target Details
| UniProt AC | P11274 |
|---|---|
| Gene Symbol | BCR |
| Protein Name | Breakpoint cluster region protein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF09036 (Bcr-Abl_Oligo) PF00168 (C2) PF19057 (PH_19) PF00620 (RhoGAP) PF00621 (RhoGEF) |
Summary
- Multi-target molecules 338
- Clinical molecules 25
- Avg pChEMBL 7.32
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (338)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KOGBNTSOPZVMIK
|
8.5 | IC50 | 2 | — | |
HXVYZZYPRMCJGZ
|
8.5 | IC50 | 2 | — | |
USIPMCNVJIUSIH
|
8.4 | IC50 | 2 | — | |
XVJQXIUEEXVEKU
|
8.4 | IC50 | 3 | — | |
ZGBAJMQHJDFTQJ
|
8.4 | IC50 | 2 | — | |
GMCVFFUTKQUYKX
|
8.4 | IC50 | 2 | — | |
HRJNCGVLSVNXDX
|
8.3 | IC50 | 2 | — | |
KWLXWXYINQHVEA
|
8.3 | IC50 | 2 | — | |
KEIRBRQKXFLPHS
|
8.3 | IC50 | 3 | — | |
XKFTZKGMDDZMJI
|
8.3 | Kd | 64 | Yes | |
FVOSLYACENHGIN
|
8.2 | IC50 | 2 | — | |
WQERLKAGPFFGAY
|
8.2 | IC50 | 2 | — | |
IZPYRHJDUKTQPR
|
8.2 | IC50 | 2 | — | |
WAFBXGBWFZZGIC
|
8.2 | IC50 | 3 | — | |
AKFZSHPZKXBMCK
|
8.1 | IC50 | 2 | — | |
NYUZAHPHSBKPPK
|
8.1 | IC50 | 3 | — | |
PJGIZSKNZNTQMF
|
8.1 | IC50 | 2 | — | |
FEYMWTKZTZABTA
|
8.1 | IC50 | 2 | — | |
UBPYILGKFZZVDX
|
8.1 | IC50 | 130 | Yes | |
BNIPBKFCGMYCDD
|
8.1 | IC50 | 2 | — | |
MNBNPSZPKJMKII
|
8.1 | IC50 | 2 | — | |
RCMBBRKIGQGXGS
|
8.1 | IC50 | 2 | — | |
REKRJPDVODUIMJ
|
8.1 | IC50 | 2 | — | |
ZGBAJMQHJDFTQJ
|
8.0 | IC50 | 15 | — | |
CGMQSJXTBXHOTH
|
8.0 | IC50 | 9 | — | |
NRSRGKSRBDKZAU
|
8.0 | IC50 | 2 | — | |
TWGQYAXRDILACQ
|
8.0 | IC50 | 2 | — | |
WXLDRYNTEQUKFN
|
8.0 | IC50 | 2 | — | |
KUNOALCWXLLCES
|
8.0 | IC50 | 2 | — | |
LCVIRAZGMYMNNT
|
8.0 | Kd | 20 | — | |
LWGSLBQDPISOIG
|
8.0 | IC50 | 2 | — | |
RZHUMJSINYZTBK
|
8.0 | IC50 | 2 | — | |
MWUBHDHHMFIRMG
|
7.9 | IC50 | 2 | — | |
SAYPRYYFORNPCK
|
7.9 | IC50 | 2 | — | |
FVYMRGNWPDZIDO
|
7.9 | IC50 | 2 | — | |
DKZYXHCYPUVGAF
|
7.8 | Kd | 112 | — | |
IHYVCWMRZWUYDY
|
7.8 | IC50 | 2 | — | |
ZGJPEVGMGPUSJY
|
7.8 | IC50 | 2 | — | |
VASBUQQNBORQFF
|
7.8 | IC50 | 2 | — | |
WHTLLTQCEBVRBM
|
7.8 | IC50 | 2 | — | |
ABIOEYXBRUITSN
|
7.8 | IC50 | 2 | — | |
KCPUHXYDPHVBQZ
|
7.8 | IC50 | 2 | — | |
LAVCQCXXKFSGQN
|
7.8 | IC50 | 2 | — | |
OUKYUETWWIPKQR
|
7.8 | Kd | 31 | Yes | |
DECSMGXZYHHMMF
|
7.8 | IC50 | 2 | — | |
LDGJWNZFGYFENB
|
7.8 | IC50 | 2 | — | |
NKEZCSVNPKYVIB
|
7.8 | IC50 | 2 | — | |
SUNRRXUOOBKXTB
|
7.8 | IC50 | 2 | — | |
ZBNZXTGUTAYRHI
|
7.8 | IC50 | 102 | Yes | |
BJCJYEYYYGBROF
|
7.8 | IC50 | 4 | — |