Target Details
| UniProt AC | P11274 |
|---|---|
| Gene Symbol | BCR |
| Protein Name | Breakpoint cluster region protein |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF09036 (Bcr-Abl_Oligo) PF00168 (C2) PF19057 (PH_19) PF00620 (RhoGAP) PF00621 (RhoGEF) |
Summary
- Multi-target molecules 338
- Clinical molecules 25
- Avg pChEMBL 7.32
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (338)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CZHIVNNGAXNFBN
|
9.8 | Kd | 3 | — | |
OHGOKRHLLKPKJK
|
9.8 | Kd | 3 | — | |
RBQXHLBIJMHVHI
|
9.7 | Kd | 3 | — | |
FGTNRYWAENEKJL
|
9.6 | Kd | 3 | — | |
KVDHKHPORALHHP
|
9.6 | Kd | 3 | — | |
IGTIROPAMADUPR
|
9.5 | IC50 | 2 | — | |
UDTHXJUPBYEYMC
|
9.4 | IC50 | 2 | — | |
YDHFUBCYRHHRFM
|
9.4 | IC50 | 2 | — | |
GNOXITMWGVMUID
|
9.4 | Kd | 3 | — | |
SRUDWIBMRKZRQG
|
9.4 | IC50 | 2 | — | |
JBMSSKLUVBBAHN
|
9.4 | Kd | 3 | — | |
OHFRVFUEGWQWTA
|
9.3 | IC50 | 2 | — | |
VOVZXURTCKPRDQ
|
9.3 | Kd | 2 | — | |
WKTHEPAGRCQCOF
|
9.3 | IC50 | 2 | — | |
AXCUTSXYMWKWEA
|
9.3 | IC50 | 2 | — | |
KOIRZEHURFRWOY
|
9.3 | IC50 | 2 | — | |
WKTHEPAGRCQCOF
|
9.3 | IC50 | 2 | — | |
WTEAUFXGRKOZNT
|
9.3 | IC50 | 2 | — | |
XJPZWFIHWISMOH
|
9.3 | IC50 | 2 | — | |
LFLRMYZNGFXKMP
|
9.3 | IC50 | 2 | — | |
LQBDBQSMCXTVKB
|
9.2 | IC50 | 2 | — | |
MQXNKLLRIGGEOE
|
9.2 | Kd | 3 | — | |
JGXRYYVIMAYABB
|
9.2 | IC50 | 2 | — | |
MKHTUOFMIYFSEP
|
9.2 | Kd | 3 | — | |
WHTDVCOWKCEOHS
|
9.2 | IC50 | 2 | — | |
ZVLDJWAUCMOGIZ
|
9.1 | IC50 | 2 | — | |
ZLMYOQZUWFEOHX
|
9.1 | IC50 | 2 | — | |
ZQOBVMHBVWNVBG
|
9.1 | IC50 | 2 | — | |
VGHMNDGFXSTBOE
|
9.0 | Kd | 3 | — | |
NUTAFQYFQXUSOF
|
9.0 | IC50 | 2 | — | |
AQSSMEORRLJZLU
|
9.0 | Kd | 34 | Yes | |
BNRXMSGHPVYSDK
|
9.0 | IC50 | 24 | — | |
QZGWWTNGPOKJGC
|
9.0 | IC50 | 2 | — | |
YLGBXIFLTCUQDE
|
9.0 | IC50 | 2 | — | |
GOEIHELWQGXKOI
|
9.0 | IC50 | 2 | — | |
PHXJVRSECIGDHY
|
9.0 | IC50 | 59 | — | |
KJOGLHQXZFOMRY
|
8.9 | IC50 | 2 | — | |
DUPWHXBITIZIKZ
|
8.9 | IC50 | 2 | — | |
SZNYUUZOQHNEKB
|
8.9 | IC50 | 7 | — | |
IQSSNBZGOCNVDV
|
8.8 | IC50 | 2 | — | |
KJIJJDDZGNJZBA
|
8.8 | IC50 | 2 | — | |
PPBMKPYHIGDXNE
|
8.8 | IC50 | 2 | — | |
UOVRWDKWWSPLGT
|
8.7 | IC50 | 2 | — | |
VAARYSWULJUGST
|
8.7 | IC50 | 119 | Yes | |
KGUOPPORYLAEOV
|
8.7 | IC50 | 2 | — | |
NFLXEOXSZWSZGF
|
8.6 | IC50 | 2 | — | |
XVCPZFLMAOLHQX
|
8.6 | IC50 | 2 | — | |
XKCPEVHEMILVAL
|
8.6 | IC50 | 2 | — | |
ALKJNCZNEOTEMP
|
8.5 | Kd | 55 | — | |
WFRLFWGASBLYTC
|
8.5 | IC50 | 15 | Yes |