Target Details
UniProt ACP11229
Gene SymbolCHRM1
Protein NameMuscarinic acetylcholine receptor M1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,571
  • Clinical molecules 35
  • Avg pChEMBL 7.27
Top Co-occurrence Targets
Active Molecules (1,571)
InChIKey pChEMBL Type Targets Clinical
SIYFJBSSISWOBJ 7.8 Ki 2
UCBXWLPRAVDTBU 7.8 Ki 5
UNZBDOQVZFAUNP 7.8 Ki 5
YPRMCONKNHLNEC 7.8 Ki 3
HBLWDHBKUANPEG 7.8 IC50 5
DRCBVHVCMKPDSV 7.8 Ki 2
DYANBEYXYZKCOS 7.8 IC50 3
FPBBKOFNQVUXDJ 7.8 IC50 3
FPBBKOFNQVUXDJ 7.8 IC50 3
IHMRJXQCYGVPPW 7.8 IC50 3
JDCADUVEQJRIDC 7.8 Ki 5
KKGVQDYTWPYXJH 7.8 Ki 3
MTBIBWFHYCAYTO 7.8 Ki 2
XPXPKUQRUOKHFD 7.8 Ki 5
JFEFOFYHVIMFRD 7.8 Kd 3
MEAOYGFCVURJIU 7.8 Kd 5
NAXYIWZRBXAQKX 7.8 IC50 3
NAXYIWZRBXAQKX 7.8 IC50 3
NGKTYFBTWFLIRS 7.8 Ki 4
QDDPQJCCXUPHKY 7.8 Ki 2
UBGMVJXVELKNMU 7.8 Ki 5
XUENORREMLOMPD 7.8 Ki 5
KKEGQSSUXOGEAF 7.8 Ki 5
NEUSVAOJNUQRTM 7.8 IC50 13 Yes
DOPPWUHKJURUAH 7.8 Ki 2
DZSCHRPHQBQAFZ 7.8 IC50 5
OHEDKBMQRCAABJ 7.8 IC50 6
DKVRRZMTJBDMTP 7.8 IC50 3
OJNGNVWCSYYTTM 7.8 Ki 2
HDOZVRUNCMBHFH 7.7 Ki 26 Yes
KYIGOCCCBXRHNJ 7.7 IC50 43
OMOWOTRKFFNAIT 7.7 IC50 5
PHTUQLWOUWZIMZ 7.7 Ki 7
VODYLGKYBHYDON 7.7 Ki 3
XRWFEGDYDKMREJ 7.7 Ki 3
DIDYGLSKVUKRRP 7.7 Ki 5
HVRWHBXGKRCKSP 7.7 IC50 3
KDASCRGXYKRCDD 7.7 Ki 3
ONSBLCCSCRKRKU 7.7 Ki 3
XBBANBCTQDQYBC 7.7 Ki 4
YECZUVJTDYORCB 7.7 Ki 3
ZWZGWXZGAUJLHN 7.7 Ki 3
BRMKEVBAZDNRPY 7.7 Kd 5
VPWKHNIBDCHPNN 7.7 Ki 5
ZMCUJOGARKOVLZ 7.7 Ki 3
HECAWZFPXYNICY 7.7 Ki 5
JCBGAEQLPPOPDK 7.7 Ki 5
OPZQMZXXMIXWON 7.7 Ki 2
RMHMFHUVIITRHF 7.7 Ki 5
SUDQOGCFXPWVPJ 7.7 IC50 4
2D structure