Target Details
UniProt ACP11229
Gene SymbolCHRM1
Protein NameMuscarinic acetylcholine receptor M1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,571
  • Clinical molecules 35
  • Avg pChEMBL 7.27
Top Co-occurrence Targets
Active Molecules (1,571)
InChIKey pChEMBL Type Targets Clinical
HTYJHPPHBQRXGX 8.1 Ki 5
PULJCGFLKSMODH 8.1 Ki 5
AVNRDCQRRUOTCC 8.0 Ki 5
KLQQZEIBZUZRLW 8.0 Ki 3
XJQLVERVBPRFET 8.0 IC50 3
XOZKVVSXDCLNPX 8.0 Ki 3
UFSZYKLBZJNXLV 8.0 Ki 5
PBHNZQQGQQOYNM 8.0 IC50 5
UACRHRRJJCXGPC 8.0 Ki 5
JATHATTURQLZHF 8.0 Ki 2
PSFULERNVNPNAD 8.0 IC50 3
XPXPKUQRUOKHFD 8.0 Ki 5
CLKYBOTWHCENMP 8.0 Ki 5
CNXWAYYAICBSCA 8.0 IC50 3
KHJKTXKHUACAIJ 8.0 Ki 5
KVWDHTXUZHCGIO 8.0 Ki 32 Yes
SLVMESMUVMCQIY 8.0 Ki 14
UNZBDOQVZFAUNP 8.0 Ki 5
DWUMIEZPQFLMBC 8.0 Ki 2
MHNSOBBJZCWUGS 8.0 Ki 17
YHOBTARVXRPKOX 8.0 Ki 4
ZMDWHSSHCTZQTD 8.0 Ki 5
AZBTYTBTYGPQFW 8.0 Ki 2
BZHQFTZHZVTIMQ 8.0 Ki 5
DFTFGLPAHCOAEP 8.0 Ki 3
GZXQKCMKEJCSMK 8.0 Kd 5
IJTZAYDMPFOINP 8.0 Ki 2
JYKJJNTVFIWSHT 8.0 Kd 5
ODAGWGUCKWUZTJ 8.0 Ki 3
SQVWTVHVWIHOSU 8.0 Ki 5
UXRUOZRDTXTVAI 8.0 Ki 5
ZUHDKSXKMLQBAW 8.0 Ki 3
AZYYVQIBCPFAIG 7.9 Kd 5
MHNSOBBJZCWUGS 7.9 Ki 3
QGJWMGIPVUWDAK 7.9 Ki 5
SPWGJUOMJHFGMM 7.9 Ki 2
FNNCHHONWUGPND 7.9 IC50 5
AYFAGRAOJPSHSH 7.9 Ki 19
YFWMVRIRFFWDJL 7.9 Ki 5
YKESQPGCPVQXIU 7.9 Ki 3
MMJNDRSEERCWAQ 7.9 IC50 3
GPFBOILGPPNQAT 7.9 Ki 4
TXAYFVDVTWJOOE 7.9 IC50 3
OIZGGNJJLMUGKL 7.9 IC50 2
SLFGIOIONGJGRT 7.9 Ki 12
NTXIFNZVYVWYBG 7.9 IC50 3
RRBQMQSYNDZVOX 7.9 IC50 3
USWIIRIGMDFSNJ 7.9 IC50 5
WHZBQLWHOPDIPC 7.9 Ki 5
NNUZSHSDIMQZLW 7.9 IC50 3
2D structure