Target Details
UniProt ACP11229
Gene SymbolCHRM1
Protein NameMuscarinic acetylcholine receptor M1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,571
  • Clinical molecules 35
  • Avg pChEMBL 7.27
Top Co-occurrence Targets
Active Molecules (1,571)
InChIKey pChEMBL Type Targets Clinical
QZQDZBWQUNVCFF 8.3 Ki 5
UFSZYKLBZJNXLV 8.3 Ki 5
XWGIZMOOTLOFBG 8.3 IC50 2
NANQRVOKMXDMNL 8.3 Ki 2
RRQOIEPFLLEXMG 8.3 Ki 3
ZVVYAPAWNNSOSQ 8.3 Ki 3
PCEDEEWEONTUHP 8.3 Kd 5
HXGBXQDTNZMWGS 8.3 Ki 8
FZXSXMYFIZKXPT 8.2 Ki 12
MDTGYTUAMOVSAG 8.2 Ki 2
SCCICKWCGZZTCM 8.2 IC50 3
UPPMZCXMQRVMME 8.2 IC50 7
CWHBWBZGFMIKAF 8.2 Ki 3
WOMCGBFNBSIIEA 8.2 Kd 5
APOMSSAGEAOUGO 8.2 IC50 5
AWMYFVQONDTWPK 8.2 Ki 2
BMNOFIWIZFZYES 8.2 Kd 5
PYSIAKZWZJNMNM 8.2 IC50 2
YQGXZPSEAUHNIN 8.2 Ki 4
UMNOHXLPNDJCMM 8.2 IC50 3
GPFBOILGPPNQAT 8.2 Ki 4
OIZGGNJJLMUGKL 8.2 IC50 4
QZUDBNBUXVUHMW 8.2 Ki 39 Yes
RSDOPYMFZBJHRL 8.2 Ki 5
WFXACEPWPCLBGC 8.2 Ki 4
GLGYXEJECWKSPZ 8.2 Ki 3
JQPHWWSHVFGYHV 8.2 Ki 3
OGTLDFSTCJABJV 8.2 Ki 5
YLJPQUAQAHVZQK 8.2 Ki 3
KLQQZEIBZUZRLW 8.2 Ki 4
CKABNURNABKRSF 8.2 Ki 2
ICZVKTVMHVHOQI 8.2 Ki 5
IJOGXSLRDLSTOS 8.2 Ki 3
RHKOEKGERJHNJH 8.2 IC50 3
YLKMPCDZOHNNJU 8.2 IC50 3
IPPGGAXXAKWHHQ 8.1 Kd 5
UECHFIXSINCEDW 8.1 Ki 5
KTWQAWSQSOISLN 8.1 Ki 4
OMZFQPGNVMBMTP 8.1 Ki 3
CZMLHCKAVIBNFO 8.1 Ki 2
JJCFRYNCJDLXIK 8.1 IC50 25 Yes
SADFFAQSWHTWLL 8.1 Ki 5
ZBEWUYNNNHETOS 8.1 Kd 3
AGVQGHLXLYNMSL 8.1 Ki 5
DUVRCCCAGVFLMM 8.1 IC50 3
LRYVHUGMUSRZRA 8.1 Ki 3
CRWJHTMQXCFORB 8.1 IC50 3
OBWGMKKHCLHVIE 8.1 Ki 9
VQMYCZUUGWZZTK 8.1 IC50 5
DUJZVZNVMYQVAM 8.1 Ki 3
2D structure