Target Details
UniProt ACP11229
Gene SymbolCHRM1
Protein NameMuscarinic acetylcholine receptor M1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,571
  • Clinical molecules 35
  • Avg pChEMBL 7.27
Top Co-occurrence Targets
Active Molecules (1,571)
InChIKey pChEMBL Type Targets Clinical
KLBQZWRITKRQQV 8.6 Ki 21
UMEDKGJVCBVATI 8.6 IC50 3
AVALEAUYDHXJQZ 8.6 Ki 3
OFTJLQGRWRVUFL 8.6 Ki 4
HLBJQGCUNYZLFQ 8.5 Ki 4
DLMOQVWYEFDOHH 8.5 Ki 5
GABVSGLOWYHOBW 8.5 IC50 3
JBVFPTKZYNRPII 8.5 Ki 3
VPWKHNIBDCHPNN 8.5 Ki 5
XHIQZUNDUKHSQA 8.5 IC50 3
MVFGNQQJJQEHLD 8.5 IC50 3
QCUQACXEVHRHIF 8.5 Ki 5
ZUXABONWMNSFBN 8.5 Ki 29
UFOTTYHVWBYOKX 8.5 Ki 5
YRRVEDQQANFYHX 8.5 Ki 3
FDGDUTRHLLBSNR 8.5 Ki 3
NEQYHZCZFMESJN 8.5 Ki 5
RTVAKAAPGHVGBW 8.5 Ki 5
STECJAGHUSJQJN 8.5 IC50 5
BSNRCPZANSBCBD 8.5 Ki 3
KLBQZWRITKRQQV 8.5 IC50 25 Yes
OYYDSUSKLWTMMQ 8.5 Ki 5
UJXAGMVNACHDOG 8.5 Ki 5
WOXZWDNEPKZBSN 8.5 Ki 3
PCEDEEWEONTUHP 8.4 Kd 5
GMLQVLRORNVELR 8.4 Ki 5
LCFLTSGKHHHXPL 8.4 IC50 3
LCFLTSGKHHHXPL 8.4 IC50 3
PXHIFOLPKHLYBX 8.4 Ki 5
FZSXJAWJJQIXFV 8.4 Ki 3
KFFUMWAFMBSHHP 8.4 Ki 4
MLKITGHXXPWOSH 8.4 Ki 5
SRLMLQNXERJQPS 8.4 Ki 4
OYXCACHCXKHEOC 8.4 Ki 5
IEEFWRMSEALUNN 8.4 Kd 5
VBBBAIRVFNYIBU 8.4 Ki 2
WHFTUKDGFGFLCG 8.4 Ki 3
ZLMYQVPAEPRSOY 8.4 IC50 3
GNQCCPIYKSBVEZ 8.3 IC50 3
HHXDJDWQQPSWHW 8.3 Ki 4
HTYJHPPHBQRXGX 8.3 Ki 5
OANBYDFPBWKVGI 8.3 Ki 5
WHKGYJCRLQITBW 8.3 Ki 5
WHKGYJCRLQITBW 8.3 Ki 5
WYDUSKDSKCASEF 8.3 Ki 5
WVAXSPFXHVXZHT 8.3 Ki 3
IENFGCJKCCNIMB 8.3 Kd 5
KCEZOSVHPLHUHT 8.3 Ki 3
RHWFCIJKMABLLH 8.3 IC50 3
LMGYQTFTIFUZCP 8.3 IC50 2
2D structure