Target Details
UniProt ACP11229
Gene SymbolCHRM1
Protein NameMuscarinic acetylcholine receptor M1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,571
  • Clinical molecules 35
  • Avg pChEMBL 7.27
Top Co-occurrence Targets
Active Molecules (1,571)
InChIKey pChEMBL Type Targets Clinical
AWYSEPZPTVMKBT 8.7 Ki 4
CBUABSHDAKLYKZ 8.7 Ki 3
CJGNMVAAMQAWEF 8.7 Ki 16
DIQXIWJNNCBKDZ 8.7 IC50 3
DPWACXBREFHUKJ 8.7 Ki 3
FIADGNVRKBPQEU 8.7 Ki 9
KUXJYXPGYUJWCD 8.7 Ki 3
NXGNXTJVCQAXEF 8.7 Kd 3
OEXHQOGQTVQTAT 8.7 IC50 5
ONOZLVJQXQZLPL 8.7 Ki 5
UBXUDWCOFMMEAI 8.7 Ki 5
WRRKXJXJKFCUCR 8.7 IC50 3
AKMDZGUFAAEGFX 8.7 Ki 5
AVNRDCQRRUOTCC 8.7 Ki 5
CBWGSRNEOFXWKO 8.7 IC50 3
GQDOZDXWIPGDGI 8.7 Ki 3
HEPQZYCRJHNVCR 8.7 Ki 3
LWKFTNSSJJTMGU 8.7 Ki 3
MBGKVLLSSVDNHB 8.7 Ki 3
OLZRBZLJTKELRL 8.7 Ki 4
PIBNOUQILXRVNG 8.7 Ki 5
PNLHOADYGQJVLG 8.7 IC50 3
STECJAGHUSJQJN 8.7 IC50 4
KFMIEAZKENMLEL 8.6 Ki 5
MMUOGZOUFNQXMP 8.6 Ki 5
PMNZXPJWRDBQSA 8.6 Ki 5
QFRDMVXRTJXQSC 8.6 Ki 5
AFLBGAQHDSOPKA 8.6 Ki 5
YSXKPIUOCJLQIE 8.6 Ki 5
ABRYVCKEQWCHSC 8.6 Ki 5
BNLVIXOVYRJUTA 8.6 Ki 5
CHCFFXBWNOXOJJ 8.6 IC50 3
GCRHFBFSDNBRFV 8.6 IC50 3
KTCCCXMNJFFEIS 8.6 Ki 3
MVMQESMQSYOVGV 8.6 Ki 3
ROCCLUYSPSAIDK 8.6 Ki 5
TYLFZULSDOOCRC 8.6 Ki 5
VRZIYMYSNOVVOK 8.6 IC50 3
OEXHQOGQTVQTAT 8.6 IC50 3
CANZROMYQDHYHR 8.6 Ki 2
HYOWZAANPMTHNJ 8.6 Ki 3
MGYXHBLZZIWHEY 8.6 Ki 3
MWLALRQZBOOMRW 8.6 Kd 3
WEFKYTFPJRTGKU 8.6 Kd 3
WXPNDRBBWZMPQG 8.6 Ki 28
XMVZKWJSNYQWPQ 8.6 IC50 3
CJDXHNZNBXVNIP 8.6 Ki 3
LPXIRSSTWSVBRH 8.6 IC50 3
YLWUNWHLKDVJRA 8.6 Ki 3
GZIIELZICVUEPK 8.6 Ki 5
2D structure