Target Details
UniProt ACP11229
Gene SymbolCHRM1
Protein NameMuscarinic acetylcholine receptor M1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,571
  • Clinical molecules 35
  • Avg pChEMBL 7.27
Top Co-occurrence Targets
Active Molecules (1,571)
InChIKey pChEMBL Type Targets Clinical
DTQIXKQBUYCCQM 8.9 Ki 3
OANBYDFPBWKVGI 8.9 Ki 5
XFUPPJKGZWWZGD 8.9 Ki 3
ZCGOYQXWRQDKNB 8.9 IC50 3
BEJYISOPDBBZRK 8.9 Ki 4
FUMDHGFBMAYXOX 8.9 Ki 3
HUARGKRBYXMIDE 8.9 Ki 3
IJPOIHRHFSVJOM 8.9 Ki 3
NEOMSSISKDUIHW 8.9 Ki 3
NHPBDFAJJFWJJX 8.9 Ki 2
GHHSRBSZNGGGPF 8.9 Ki 3
IEENUMOCDKBVGC 8.9 Ki 4
HWHLPVGTWGOCJO 8.9 Ki 6
DFCLHAWGKPEFIX 8.9 Ki 5
UOKGNINOAYOIDX 8.9 Ki 5
CXRIFSPGYWTKPW 8.8 IC50 3
FOJQLTRBJHZZKU 8.8 Kd 3
JNJKTGYSCZXDCF 8.8 IC50 3
LYFQHKXGGDVXCQ 8.8 Ki 5
NQWKKVJOEVKIHT 8.8 Ki 3
OOGJQPCLVADCPB 8.8 Ki 9
XFGSFWFIJFNGQY 8.8 Ki 5
DFCLHAWGKPEFIX 8.8 Ki 5
CXCOPHKFCPOFFH 8.8 Ki 3
DJOCICQNBMTMNG 8.8 Ki 5
GXQAMXKWCFMGON 8.8 Ki 3
HQRSMNLSFMUJPL 8.8 Ki 3
QRUXDRCXIGZTGT 8.8 Kd 5
URDXFKMXLZZTRI 8.8 IC50 3
ZUICJRIEMALFLN 8.8 IC50 3
XIQVNETUBQGFHX 8.8 Ki 10
CJRUIOCIHPGNQL 8.8 Ki 5
HDAMOICMOAXFLJ 8.8 Ki 4
LMDNOMYZUIYOBM 8.8 IC50 3
ULGLMVSOOWNSNJ 8.8 Ki 3
WKWYANDGYZVVAK 8.8 IC50 4
YUJOQEAGGUIMED 8.8 Ki 5
ZGAIDOGAKIQCJU 8.8 IC50 3
CURUTKGFNZGFSE 8.8 IC50 10
GKDBTHSYQZTDAJ 8.8 IC50 13
RKAJVTVMICVPJE 8.8 IC50 3
DUMGHCJXMGZUEK 8.7 Ki 3
JGOIBENTSQHWDQ 8.7 Ki 5
OWDSSIDYHAEOHU 8.7 Ki 3
PEOXDNXZHVLPEP 8.7 Ki 3
QOJBMAYEUGMTTA 8.7 Ki 5
RXLCWZMWTUZMFM 8.7 Ki 3
HPHMHCRNJVKYKE 8.7 Ki 4
POIIDLJXIAHDFT 8.7 Ki 5
ZDFAGRMEOOJZOO 8.7 Ki 3
2D structure