Target Details
| UniProt AC | P11229 |
|---|---|
| Gene Symbol | CHRM1 |
| Protein Name | Muscarinic acetylcholine receptor M1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 1,571
- Clinical molecules 35
- Avg pChEMBL 7.27
KEGG Pathways (9)
Active Molecules (1,571)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NHFIEMNGVIAFJO
|
6.0 | Ki | 3 | — | |
BKVIWGRFRKLFIO
|
6.0 | Ki | 9 | — | |
FWDQHCMQPLYEEB
|
6.0 | IC50 | 3 | — | |
HMXDWDSNPRNUKI
|
6.0 | Ki | 72 | — | |
LDMXQNXCFMLIER
|
6.0 | Ki | 2 | — | |
OEUUCWVHNBAMPM
|
6.0 | Ki | 3 | — | |
PNVNVHUZROJLTJ
|
6.0 | Ki | 6 | — | |
QCTZZHSEDPYHIV
|
6.0 | IC50 | 4 | — | |
RZSWLEFBXTVYMU
|
6.0 | Ki | 3 | — | |
SBCYNHCFJBYRJY
|
6.0 | Ki | 3 | — | |
SGVSRMZTPNFPFO
|
6.0 | IC50 | 4 | — | |
UDVBAIMSAZRJGM
|
6.0 | Ki | 2 | — | |
VHGCDTVCOLNTBX
|
6.0 | Ki | 19 | — | |
VKXFSAYDXXXNGC
|
6.0 | IC50 | 3 | — | |
VSIWWORCEGQUCZ
|
6.0 | IC50 | 3 | — | |
WUQAXDTXXDUDGH
|
6.0 | IC50 | 3 | — | |
XIVKYSIXVZBKEK
|
6.0 | Ki | 2 | — | |
XKCJLNBEKXPHNT
|
6.0 | IC50 | 3 | — | |
XKJHWFAMUVWRDJ
|
6.0 | IC50 | 3 | — | |
ZETHWWBQKDKSDJ
|
6.0 | IC50 | 3 | — | |
ZEUITGRIYCTCEM
|
6.0 | Ki | 12 | — |