Target Details
UniProt ACP11229
Gene SymbolCHRM1
Protein NameMuscarinic acetylcholine receptor M1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,571
  • Clinical molecules 35
  • Avg pChEMBL 7.27
Top Co-occurrence Targets
Active Molecules (1,571)
InChIKey pChEMBL Type Targets Clinical
ALYUIXQXWXKCQL 6.1 Ki 2
CCRWXCJNGCBNBD 6.1 Ki 2
CFUNJFPJLPERDK 6.1 IC50 4
CZKLKFHCKZAYEM 6.1 IC50 4
GVNXJWWMOLONBJ 6.1 IC50 2
MAILZJQPMMCTKE 6.1 IC50 4
RTHCYVBBDHJXIQ 6.1 Ki 15 Yes
VSOCKTWBYUTTOC 6.1 IC50 2
XQXLJONHFLRFOK 6.1 IC50 4
YYODSLJMAMEDBQ 6.1 IC50 4
GXLBEEGSWNFNGE 6.1 IC50 4
MTDYDDJVCIHZKH 6.1 Ki 7
PRGSUPYUMMZLEM 6.1 IC50 4
PWYNNAYMPKVKJL 6.1 Kd 5
RHAFROHARIZTPJ 6.1 Kd 5
AWSWSDJGJTXACL 6.1 Ki 11
COXRSODPRFBGSM 6.1 Ki 3
FJOQSAAWJBXPCK 6.1 Ki 5
KLYUNLYWGBECRC 6.1 Ki 3
MUFOTJYSFCKGKD 6.1 IC50 2
MVKKLGNVARQKRP 6.1 Ki 13
MWDWETWIXZBNRI 6.1 Ki 2
SOZIYETWMOLCLB 6.1 Ki 2
ZGQSHOMCFXQQCY 6.1 IC50 2
ZYBBUFPKZJQNLL 6.1 Ki 3
AFNXATANNDIXLG 6.0 Ki 11
ANTKBACNWQHQJE 6.0 Ki 12 Yes
GWWHCPBYLSKMJU 6.0 Ki 3
HDUFNCWFVWHJPJ 6.0 IC50 3
HYKCKUKATCYSMY 6.0 IC50 2
LFSUTWJOQHTMTB 6.0 IC50 3
OMYFTZZTQULVGM 6.0 Ki 2
SBWDNXAOTCMVAA 6.0 IC50 7
KKLOVGWFIDGYBH 6.0 IC50 4
LNSFWYTUQPZOOX 6.0 IC50 4
SRADGLKKIKVDBB 6.0 Ki 2
VMJSEWCRPGCNOF 6.0 Ki 5
YEWCXJGTKBDZNL 6.0 Ki 2
BHNWCPXBMCJVAS 6.0 Ki 5
GPZMWOXSIRVXQW 6.0 Ki 8
MCVGJQYUOLRXOM 6.0 Ki 3
QFUMICBVJQFZRC 6.0 IC50 4
BYBLEWFAAKGYCD 6.0 Ki 16 Yes
CCMKPZZOFUAWCG 6.0 IC50 3
DZPZVLKXEXASCW 6.0 IC50 2
NJFIHVYKGVSISN 6.0 IC50 4
PCWGGOVOEWHPMG 6.0 Ki 12
SNWLCKAUHVWOLQ 6.0 IC50 4
UKHHETYTQCSWPT 6.0 IC50 2
MITFBVJTVLMZJU 6.0 Ki 2
2D structure