Target Details
UniProt ACP11229
Gene SymbolCHRM1
Protein NameMuscarinic acetylcholine receptor M1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,571
  • Clinical molecules 35
  • Avg pChEMBL 7.27
Top Co-occurrence Targets
Active Molecules (1,571)
InChIKey pChEMBL Type Targets Clinical
JKGARLBCOXRROD 6.2 Ki 5
SMANXXCATUTDDT 6.2 Ki 25 Yes
DATRLTNBZWRBPI 6.1 Ki 12
HJWZLXLUSXAXBS 6.1 IC50 4
KLFGFVJTTRHXMN 6.1 Ki 2
PEBPHJVYNJHNAS 6.1 IC50 4
VAIOZOCLKVMIMN 6.1 Ki 3
VICTYDRNEFPKTN 6.1 Ki 5
AAPXNHMQKBDDJN 6.1 Ki 4
CNDOHBNSSCZYEQ 6.1 IC50 2
CNDOHBNSSCZYEQ 6.1 IC50 2
HAUISRCENQSVAD 6.1 IC50 4
HBRHULDGKNIFGB 6.1 Ki 4
JMEYTJRRQTXEIE 6.1 IC50 4
MCGDBHZRFQKLBT 6.1 Ki 3
RPWGPUBKJDYNDR 6.1 Ki 2
YBHILYKTIRIUTE 6.1 Ki 11
ZRESSCFPNIPPGT 6.1 IC50 3
FGWDVBIHPBYKJI 6.1 Ki 2
HKRMWBKEZJIJNK 6.1 IC50 3
HLFXMJFGYOOILI 6.1 Ki 3
JRTMAXYLOBYIGG 6.1 Ki 2
WMHFTJFIHGBUHI 6.1 IC50 4
BDKHSETYUSIWLB 6.1 Ki 3
KYIAOTGZEXVAKQ 6.1 Ki 2
LVAXIKIVPNIRLY 6.1 IC50 2
LXHDJDGOVRXFAY 6.1 Ki 2
RTHCYVBBDHJXIQ 6.1 Ki 15
TTWJVFZECWBGRO 6.1 IC50 4
ANUNMVJZPWGZDH 6.1 Ki 5
DKHZVOWFKMHNPB 6.1 IC50 3
DUYRWEBTZNUILI 6.1 IC50 4
GUYHTHYSWVZNOT 6.1 Ki 3
IMKYINSUEJXTJZ 6.1 Ki 5
JRUSYSCSOBAJQG 6.1 Ki 5
KRNTULKYNGVTDS 6.1 IC50 4
LUXQIYXMOWBLGG 6.1 IC50 4
WRWFIBSHOMVGDI 6.1 Ki 2
XNEGPONSGSBZSW 6.1 Ki 3
ZZLXMAVIXOPGOF 6.1 IC50 4
BURCDLIOLMBANF 6.1 IC50 2
JMUXXPVTXZBUDS 6.1 Ki 2
RXJJLNUPBMTGAW 6.1 Ki 5
RXJJLNUPBMTGAW 6.1 Ki 5
SKJCFKSSJBSZHL 6.1 IC50 4
SPKUCVZRLVPSOG 6.1 IC50 4
VLPCMABIYZTMKT 6.1 Ki 2
XTDVAENSULGVTJ 6.1 Ki 5
YIQPUIGJQJDJOS 6.1 Ki 5
ABOBMBIQQPJTMJ 6.1 IC50 5
2D structure