Target Details
UniProt ACP11229
Gene SymbolCHRM1
Protein NameMuscarinic acetylcholine receptor M1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,571
  • Clinical molecules 35
  • Avg pChEMBL 7.27
Top Co-occurrence Targets
Active Molecules (1,571)
InChIKey pChEMBL Type Targets Clinical
CZTMYBUHNDAZEH 9.1 IC50 3
KKEGQSSUXOGEAF 9.1 Ki 5
KWNNFRFNOLSRJT 9.1 Kd 3
SRSDGJOKLMADHL 9.1 IC50 3
UOKGNINOAYOIDX 9.1 Ki 5
XJFLDBYRKJAMIK 9.1 Ki 5
MTYMLJSBEPCLGC 9.1 IC50 3
PHRZGNXUUFTVSE 9.1 Ki 5
PHRZGNXUUFTVSE 9.1 Ki 5
OEXHQOGQTVQTAT 9.1 Ki 5
PHCOXGCMPCMSJB 9.1 Ki 3
KOKXORZIPKJNJL 9.1 Ki 5
ZHLYDKYZZGUNHA 9.1 Ki 3
RKUNBYITZUJHSG 9.1 Ki 7
UXZDMXYRRQJIBJ 9.1 IC50 3
ZJSWMRJWTWJORH 9.1 IC50 3
DFCLHAWGKPEFIX 9.0 Ki 5
VQESBLKWYKQKCC 9.0 Ki 3
VMRVZDOCRVNUDB 9.0 Ki 3
ZLCXSBBNUIIBRK 9.0 Ki 3
WCMVSMOIDILBOJ 9.0 Ki 5
ZAJRAXXUFDGAST 9.0 Ki 3
ZZCCWXNFFGHRJX 9.0 Ki 5
INNRKNITHWITSQ 9.0 Ki 3
CFPVEUFKLQKJRS 9.0 IC50 3
FTPFTSZCIOVABV 9.0 Kd 3
KZJQTCGYGSMOSC 9.0 IC50 3
LLPYCIXHQOFZRV 9.0 IC50 3
NAOXUXMOYDUMFJ 9.0 Kd 3
PFSPMYHTZUFJQW 9.0 Ki 5
QJBDLOQOXGQJTD 9.0 Ki 5
URMUNPDVNSULQI 9.0 Ki 3
WRQCVLFZYUVEBT 9.0 IC50 3
CNWBYOPCIWGBPG 9.0 IC50 3
CTMFSRXCRWGXJY 9.0 Ki 3
HYJRTXSYDAFGJK 9.0 Ki 5
JXUDJJIKYUMXJI 9.0 Ki 3
LIAJJEHSFRHBLC 9.0 IC50 3
NCPVINAZNPBCKE 9.0 Ki 5
CHLSHLSJSIBNQZ 8.9 Kd 3
GKEOHNSBCHXZOA 8.9 Ki 3
MNGBIMWSQDCYMU 8.9 Ki 3
UCURTLDVWIWPRM 8.9 Ki 5
WXIPHGJGJFDRNH 8.9 IC50 3
INEDRTXKDAPQKU 8.9 Ki 5
SRNHSTWHMJIPBN 8.9 Ki 3
LISJYMSYSGWFLD 8.9 Ki 5
MVNBPMNELMRFMU 8.9 Ki 5
MVNBPMNELMRFMU 8.9 Ki 5
AKPOTJIMZXGFLY 8.9 Ki 5
2D structure