Target Details
UniProt ACP11229
Gene SymbolCHRM1
Protein NameMuscarinic acetylcholine receptor M1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,571
  • Clinical molecules 35
  • Avg pChEMBL 7.27
Top Co-occurrence Targets
Active Molecules (1,571)
InChIKey pChEMBL Type Targets Clinical
PFQNHVGTLFNXFJ 6.3 Ki 4
PNUJBDRLVYCHKZ 6.3 Ki 2
PPVUGQCZCVNEJQ 6.3 Ki 3
QDMNOCJCRKNVJN 6.3 IC50 4
QESPLEGLQLFXGC 6.3 Ki 3
QGFRSCCIOLHNLP 6.3 Ki 2
QIRMACDSTYNSCC 6.3 Ki 2
QLHPXZICVIHDES 6.3 Ki 4
QLVPZVQOSYIUDP 6.3 Ki 2
QTHLDHUQZSKBDD 6.3 Ki 2
RLTFQBBUOILINJ 6.3 Ki 3
RQUSADBDDUGFKK 6.3 Ki 3
RXSNACAZEYSDGE 6.3 Ki 3
SBNZJHZLEKUKOR 6.3 Ki 2
SMFZJNAQVMLPNH 6.3 Ki 2
SPKCOBCJOCXPSR 6.3 Ki 2
UGMRMSCESDAAEU 6.3 Ki 2
UNJWATOCEVODBR 6.3 Ki 2
UNJWATOCEVODBR 6.3 Ki 2
UPQFMOHGVPABFY 6.3 Ki 3
VJPSKBYMCHVXKK 6.3 Ki 2
WCOCCFQTXCRQFR 6.3 Ki 3
WYBKOFUVDMJWMJ 6.3 Ki 2
XAONVLSEMXSGTB 6.3 Ki 2
XRXXVCCJOHONHF 6.3 Ki 3
XVNPANUOICOMOG 6.3 Ki 2
YSKBYDHKCWCHNB 6.3 Ki 2
YWBLUYIJHOWRBA 6.3 Ki 4
ZEJFPLCAHPOHAH 6.3 Ki 2
ZJYJBYLPHGQXEJ 6.3 Ki 3
LRMWMKQIJLOEPF 6.2 Ki 3
NKHWHVPIQQFKIT 6.2 IC50 4
PAJSQNJPMJTKTN 6.2 IC50 6
SEVOIKJSSMTXNE 6.2 Ki 3
TWMKVARMUAJVEO 6.2 Ki 2
AOYBULVQHCLRGS 6.2 Ki 3
CBDJZHFJKQNGLM 6.2 Ki 5
FWVRMDGONFOSIW 6.2 Ki 5
HMBFXHIQISYDKM 6.2 Ki 4
RSMOYRFTQUYBTP 6.2 Ki 5
TWZHATSAMULYRA 6.2 Ki 2
UECJYWWGFQYNFJ 6.2 Kd 5
WEHSOOUZRJEYJK 6.2 Ki 2
HWEGXFSUSOJEQJ 6.2 Ki 3
VDJFLDNOQKUSKT 6.2 IC50 4
VIXVIRHYJPIXPC 6.2 IC50 3
ABFWCAYAWMISPA 6.2 IC50 3
BRBVBRCNTVSDRI 6.2 Ki 2
CCQBBHNLKQFRRR 6.2 Ki 3
DERZBLKQOCDDDZ 6.2 Ki 20 Yes
2D structure