Target Details
UniProt ACP11229
Gene SymbolCHRM1
Protein NameMuscarinic acetylcholine receptor M1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,571
  • Clinical molecules 35
  • Avg pChEMBL 7.27
Top Co-occurrence Targets
Active Molecules (1,571)
InChIKey pChEMBL Type Targets Clinical
MHPRRIFCBPETQG 6.3 IC50 3
OALBGXZFCMPEGE 6.3 Ki 3
QWECGXAFJUBHNJ 6.3 Ki 2
SZXDNUASCUAYNA 6.3 Ki 4
UGIKUWKKYSFRTQ 6.3 Ki 2
XTZMDCZEQAAHDQ 6.3 IC50 4
YTQOJNIHNFXEJR 6.3 IC50 4
AFAZXESEAHMGAC 6.3 Ki 4
AMKGONWYZZPTIL 6.3 IC50 4
DGRHJZMAQQIHDX 6.3 Ki 5
DLICIVPXYFTRLA 6.3 IC50 4
HCVAFIOQGLGPAZ 6.3 Ki 5
KVDGLEHCVWVBQY 6.3 IC50 3
PZIGTEKDSRHYIT 6.3 IC50 4
FJUJIAPJEKDAAL 6.3 Ki 2
PGZUAZYZPAOAOH 6.3 Ki 2
QAZOBYCWYDQBSG 6.3 IC50 2
RYYQFPBFNFAVFQ 6.3 IC50 4
SQSAXGWIZUBYJD 6.3 Ki 2
ATMXUFMBNANYLL 6.3 Ki 5
LRBPZOOGQFAYKA 6.3 Kd 5
MNAFRWGRFIBAQX 6.3 Ki 4
NBHKBEGQNUWGRE 6.3 IC50 2
RNRYJWQFMOEPCM 6.3 IC50 2
VIEHHRQCEMIKCL 6.3 Ki 2
AJNMOHQSPDQJMZ 6.3 IC50 4
DQNCRNVCBHYBQP 6.3 IC50 4
QFWVGKDFYOXTQO 6.3 Ki 4
XJTVRXYTOLNCDQ 6.3 Ki 4
YTJBCMWEQPWTAA 6.3 Ki 6
AVBKRVFZNFJQBK 6.3 IC50 3
BOIBFMBXKXOTTH 6.3 IC50 4
CDKSQJVFQYAHGP 6.3 IC50 4
CTPZAQGPYTYXAV 6.3 Kd 5
FPDIERBPQFAFSI 6.3 Ki 17 Yes
JKVQLYYFJAJPMT 6.3 IC50 4
LJYNEMRCASTSJC 6.3 IC50 3
NPKXLQFZQRGXGC 6.3 IC50 4
DNTMJQSPHMJSNX 6.3 IC50 4
FIYZCZVBIXLYNG 6.3 IC50 3
GEKJAYDKEVECQC 6.3 IC50 2
HPXSCBIGYJMQQH 6.3 Ki 5
HVYLLNOLIBCXLL 6.3 Ki 2
KBFDMWOMIBRCFI 6.3 Ki 2
NHUMNXSOVZCLNK 6.3 Ki 11
PNEQLTWPDVHRRF 6.3 IC50 3
WEEBXSDEOQNZPK 6.3 Ki 3
WLFNSLXDBGXUSV 6.3 IC50 4
HHDGJFBTFPNSEV 6.3 Ki 5
UNOFGQWDNLJPIO 6.3 Ki 2
2D structure