Target Details
UniProt ACP11229
Gene SymbolCHRM1
Protein NameMuscarinic acetylcholine receptor M1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,571
  • Clinical molecules 35
  • Avg pChEMBL 7.27
Top Co-occurrence Targets
Active Molecules (1,571)
InChIKey pChEMBL Type Targets Clinical
STIWHEMFVTWALB 6.4 Ki 5
ZBZJUNCNHQXSBX 6.4 IC50 4
GKIRPKYJQBWNGO 6.4 Ki 20 Yes
LRMWMKQIJLOEPF 6.4 Ki 2
ADHSKYZRIOAFEG 6.4 Ki 2
HSFWTAVXXXJJRW 6.4 IC50 2
MQFKIDUREUWWAN 6.4 IC50 2
NQBVJJZTZVZQNO 6.4 IC50 4
PGDYOGMNQCUWMZ 6.4 Ki 5
QQJHRQZZCNYDMX 6.4 Ki 11
UMJCXNQRGMBWAP 6.4 IC50 4
XARSDFQMNNNPBL 6.4 IC50 2
CSFZKHHTENQXJK 6.4 Ki 2
GESNBHIZDFFLSC 6.4 IC50 4
JXWRUAABQDEVFS 6.4 IC50 4
MAFMKKCYGMIRLR 6.4 IC50 4
NNDGJLSCEUBTOL 6.4 IC50 4
PAYAQSDGYIQGSL 6.4 Ki 2
SFLBUYYNIAMYCQ 6.4 IC50 4
AIECXAGTKDCJRA 6.4 IC50 3
BZIDQKPJJVZXGZ 6.4 IC50 4
BZWYVCIHWVRXMT 6.4 IC50 4
CEOPDYXKQNAOAS 6.4 IC50 4
CHSDYWULPTYCTA 6.4 Kd 5
KEEHNWJFNGQLMW 6.4 Ki 2
RBFJBYJDTRIQFT 6.4 IC50 4
UOAPPNMLTJVXDT 6.4 IC50 4
WUPKEZLEBLCZJB 6.4 Ki 2
XBJVFFSOHGDXIL 6.4 IC50 3
XJLOQWKHCAZUQM 6.4 Ki 2
XJLOQWKHCAZUQM 6.4 Ki 2
ANBSDISLLOPZAN 6.4 Ki 2
DFWUAFCLJJBUNR 6.4 IC50 2
FMPNFDSPHNUFOS 6.4 Ki 3
HDXVOMCKOIYVCK 6.4 IC50 4
QCTSRLYZXNHQPV 6.4 IC50 2
RLUNJKJUFRFYJM 6.4 Ki 4
VGKDLMBJGBXTGI 6.4 Ki 7
WQEUCWAEHCWTPL 6.4 Ki 3
YKMYFJKVCCQVAY 6.4 Ki 2
ZRJDXADSUVEXJL 6.4 IC50 4
ZUSQEIFGHOIMSY 6.4 Ki 5
BKLZRBBUIURTRR 6.4 IC50 4
LGCNGBKZRRQUBB 6.4 Ki 5
OIYSCQVQNFKYTO 6.4 Ki 2
OIYSCQVQNFKYTO 6.4 Ki 2
QDYDEMPAIUGHBP 6.4 IC50 4
YSPKJODQLIOHOF 6.4 Kd 5
ZVIPUTDHIIGPSP 6.4 IC50 4
HTICRTTUUTUNSK 6.3 IC50 4
2D structure