Target Details
UniProt ACP11229
Gene SymbolCHRM1
Protein NameMuscarinic acetylcholine receptor M1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,571
  • Clinical molecules 35
  • Avg pChEMBL 7.27
Top Co-occurrence Targets
Active Molecules (1,571)
InChIKey pChEMBL Type Targets Clinical
PJYMPYZYAUFCMF 6.5 Ki 3
SOYKEARSMXGVTM 6.5 Ki 8
UVKZSORBKUEBAZ 6.5 IC50 13 Yes
HOFRPDJMFZKVCV 6.5 IC50 4
JLVFDXYWPHSZHA 6.5 IC50 4
JMEYTJRRQTXEIE 6.5 IC50 4
LBMILISNRUJASD 6.5 Ki 2
NUJWKQSEJDYCDB 6.5 Ki 4
PQLJILRFRUEHRW 6.5 Ki 2
SWFSQSZMVIJILA 6.5 Ki 3
WBJWKXMRVRYDQU 6.5 IC50 4
WZYQNTPWCRAGPJ 6.5 Ki 2
BGECMWFZHVFBGB 6.5 IC50 3
GQTREADDTJPDTG 6.5 IC50 4
HNQCDUJRXDPLHW 6.5 Ki 5
IACKPEHSXQAEKP 6.5 IC50 4
LQOJFNRTYZDTBR 6.5 Ki 5
QDGDDAFKQVQWCI 6.5 Ki 5
RQDGBNLSKUOAJD 6.5 Ki 3
UEQUQVLFIPOEMF 6.5 Ki 21 Yes
WMGWWIZDKKAUOR 6.5 Ki 3
FRSBYJSARNVZCX 6.5 Ki 5
IOQZWNCABFVBOY 6.5 Ki 2
QCSKQMQBRQOXLU 6.5 Ki 5
QHFVUCATFKHMCG 6.5 Ki 5
WOWRXMYCLGLRFQ 6.5 Ki 7
BJUQLFXRXSMDCM 6.4 Ki 5
GCMYOOAJYOMGJH 6.4 Ki 5
JYSMOALYFDOUBL 6.4 Ki 3
KWJYQGYMUAXZAM 6.4 IC50 4
MYQTVOSXIIRICR 6.4 Ki 5
VNTBTHFURNKMMY 6.4 IC50 4
YCGXHEJETHPGPD 6.4 Ki 8
ZXMNYBKMHVSGDY 6.4 IC50 4
AWEBVNCNTLOVSN 6.4 IC50 5
FPGYVSKEOKZERL 6.4 Ki 5
JGTJANXYSNVLMQ 6.4 Ki 2
MUCSIJXVXPLNPT 6.4 IC50 4
OMUDHMBLKINCCX 6.4 Ki 3
PAXJABBAIBFJBH 6.4 Ki 4
QOECJCJVIMVJGX 6.4 Ki 8
TZADATSLTAFDKI 6.4 Ki 3
WTVQMTFZYWXSRS 6.4 Ki 4
WYXGHKGJTWRLPO 6.4 Ki 2
AWAIMVZXXQUWMW 6.4 IC50 3
BHMUJUZQLJUJEX 6.4 Ki 3
GIARMOGSIPBRHC 6.4 IC50 4
HRIDJFHKBNVJDP 6.4 Ki 5
KDTXPLWOUMFWJY 6.4 Ki 2
QJZTYRBARUHAQD 6.4 Ki 3
2D structure