Target Details
UniProt ACP11229
Gene SymbolCHRM1
Protein NameMuscarinic acetylcholine receptor M1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,571
  • Clinical molecules 35
  • Avg pChEMBL 7.27
Top Co-occurrence Targets
Active Molecules (1,571)
InChIKey pChEMBL Type Targets Clinical
SCKFVSKZQOECOJ 6.5 IC50 3
VBTYLZVMQCAWDY 6.5 Ki 4
VMFLQXFBDYJKML 6.5 IC50 2
WEVVZJGQIWKFOJ 6.5 Ki 2
XFBTXTHJTCSANR 6.5 Ki 5
ZJTPWNRJJWBBAU 6.5 IC50 4
HTKBZSOYVFEBSC 6.5 Ki 5
LTXREWYXXSTFRX 6.5 IC50 3
SHORJVPMMAZEFL 6.5 Ki 4
AIZMFPJJDXEQKC 6.5 Ki 4
CZWQBSKNHUVZLI 6.5 IC50 5
DGWWXFCHEOPTQT 6.5 Ki 3
DKABYCZEFMBXSO 6.5 Ki 4
GJETZLQENWRAAE 6.5 IC50 4
GUNNKZVYPHUUKA 6.5 IC50 4
JVGDBVAGMMZAGB 6.5 Ki 3
MVWIZZHMSROILD 6.5 Ki 4
MVWVFYHBGMAFLY 6.5 Ki 31 Yes
OJKKZNGEMBSWMR 6.5 Ki 2
PIYDQIQMOSYBMU 6.5 Ki 4
UFCZLLHJHLQHLW 6.5 IC50 4
WNQGWYNSYNFIHU 6.5 Ki 3
JQRGZCIIOMPAEJ 6.5 Ki 2
LPTBHUFJWMXONX 6.5 Ki 2
MNAFRWGRFIBAQX 6.5 Ki 6
ODSPZLQLPQOLJR 6.5 IC50 3
OEFNMCGLYOCCQF 6.5 IC50 4
VGKDLMBJGBXTGI 6.5 Ki 15
XEKLOEGUGVGFFA 6.5 IC50 4
DMFXETUOWLUQID 6.5 Ki 5
IDQNRTMGRDBENG 6.5 IC50 4
IJIHPPHWXPHTRG 6.5 IC50 2
LOAZWNRCWBWKAC 6.5 Ki 5
NWMFUMWLMFJZLH 6.5 IC50 5
OCOMTFATMRIOSP 6.5 IC50 5
WEGLOYDTDILXDA 6.5 Ki 22
WWXCWTRLUXMAHX 6.5 Ki 7
IDQDYULTECQGBI 6.5 IC50 3
KFIBFLUHCJZUTE 6.5 IC50 3
OBLWLENBNRYSCO 6.5 IC50 5
OGAKLTJNUQRZJU 6.5 Ki 9
UBGMVJXVELKNMU 6.5 Ki 5
WIEMOFKMOGPXQF 6.5 Ki 5
ZIQDGXNDXRMRPM 6.5 Ki 6
AVNRDCQRRUOTCC 6.5 Ki 4
FHPIXVHJEIZKJW 6.5 Ki 18 Yes
FTTBANDCEOHFPG 6.5 Ki 4
KQNCPMKGQUVCKN 6.5 IC50 4
NBNHGRRWKSPRMB 6.5 Ki 2
OXWXUIXTFQJYIL 6.5 Ki 5
2D structure