Target Details
UniProt ACP11229
Gene SymbolCHRM1
Protein NameMuscarinic acetylcholine receptor M1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,571
  • Clinical molecules 35
  • Avg pChEMBL 7.27
Top Co-occurrence Targets
Active Molecules (1,571)
InChIKey pChEMBL Type Targets Clinical
GCUKWJUJMLWMQG 6.7 IC50 4
IAEZSAZZZCBEAM 6.7 IC50 4
LFBDZBNSTSRAPO 6.7 IC50 4
LQFCVVPCKLVIJM 6.7 IC50 4
PLQQFQYHSIBALT 6.7 Ki 3
UPDAFPDJKSGPME 6.7 Ki 5
VHCDKYWUNQXVAJ 6.7 Ki 3
XUJYIQJVTCUDPS 6.7 IC50 4
XWZQPFIZAGITHQ 6.7 Ki 4
ZADZTHCBMHAULL 6.7 IC50 4
DDXKWKGIBLVYQU 6.7 Ki 5
JAETUXLDWVGPIH 6.7 Ki 2
JNOSYXLLGUQJNO 6.7 IC50 2
PQHIRTDXFUZNBI 6.7 Ki 5
ULAXKLBWXHXBQI 6.7 Ki 3
CTSIKYPJIHWEIY 6.6 IC50 4
DHRLTOSMTNHHKC 6.6 Ki 4
HQQZMWSGDGFMAD 6.6 IC50 4
IENZWNOPOBXYDA 6.6 Ki 4
LACUGMNHRWEZND 6.6 Ki 5
MVULQCLNWNITMJ 6.6 Ki 3
OUCWEZXREOJVEN 6.6 IC50 4
SWFSQSZMVIJILA 6.6 Ki 2
TUIVYXUOOMYSLZ 6.6 Ki 2
UOGBSPSWAMZQNS 6.6 IC50 2
VUCYYOGBXRCVIJ 6.6 Ki 5
WPNMJEWMGWUSOR 6.6 IC50 4
ZSEXCDQYDWJYHN 6.6 Ki 5
NYNKCIGJEUJVIL 6.6 IC50 2
PHMGZAICAOYEAF 6.6 IC50 9
ATALOGFLLWJSLP 6.6 Ki 2
IRMGRKYAWRQXGM 6.6 IC50 4
JDMLRAOKSMUFSO 6.6 Ki 2
JIGSPXRYDBBYSX 6.6 IC50 4
JPOYKIKTCAMMKF 6.6 IC50 4
RCPNNLKDMRCWCD 6.6 Ki 5
VHYUYQHTMPWAPK 6.6 Kd 5
VMDQJWCKNWZEFM 6.6 IC50 4
WEGLOYDTDILXDA 6.6 Ki 22
BSSWNYCCQZRJSB 6.6 Ki 5
HNLUMKGZTQUVEY 6.6 Ki 5
KQRIXGFCTRCLAY 6.6 Ki 3
WIKYUJGCLQQFNW 6.6 Ki 23 Yes
AMWYWNMCYBNFMO 6.6 IC50 3
AUHCHCMUODVFLL 6.6 Ki 2
BFELQLHLUNQIHL 6.6 Ki 3
DBTFFFQVHFURIG 6.6 IC50 4
DJBUGHJJKOXHDD 6.6 IC50 5
DOTRMAARWOGFII 6.6 IC50 3
GUPWBMMEJNAFFT 6.6 IC50 3
2D structure