Target Details
UniProt ACP11229
Gene SymbolCHRM1
Protein NameMuscarinic acetylcholine receptor M1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,571
  • Clinical molecules 35
  • Avg pChEMBL 7.27
Top Co-occurrence Targets
Active Molecules (1,571)
InChIKey pChEMBL Type Targets Clinical
PABWMVGKWJUEBB 6.8 Ki 2
QCCFFOJHBRUSTA 6.8 IC50 4
WOQRTLKHUAYKIA 6.8 IC50 2
XFRRXQDVSCYLBU 6.8 Ki 5
ZOEYTLRCDGNMCU 6.7 Ki 5
FRACQPHKPHCEIE 6.7 IC50 4
FTFRVHRVNAJZCB 6.7 Ki 3
GSTSHGWHXRRCHO 6.7 Ki 3
MVMQESMQSYOVGV 6.7 Ki 6
MVNBPMNELMRFMU 6.7 Ki 5
OIIHCBDCPNFEIZ 6.7 IC50 4
PAESGWBCWVGCNX 6.7 IC50 4
QZTQQKQHRWQZMZ 6.7 Ki 4
SOYSPNNNWBPAGF 6.7 IC50 4
UJCYUJOQBXHJFH 6.7 Ki 4
VFGCJSNSBKYESO 6.7 IC50 4
GRHQYMDSSBRZTL 6.7 Kd 5
UUQSWYMJKUSTBX 6.7 Ki 3
BPADOPKTHDTFRT 6.7 IC50 4
CAGFDMXWWOBBHR 6.7 Ki 5
DXXIKGWICQKDRH 6.7 IC50 4
HBJANPVGVPJJER 6.7 IC50 3
HLZNMIGIMIMVBL 6.7 IC50 4
IQWCBYSUUOFOMF 6.7 IC50 4
LAYPCPWQLOVMFU 6.7 Ki 3
MRTRSVIAPJHYNC 6.7 Kd 5
NBAJZOJKXOSUNZ 6.7 IC50 2
OJFDFZDJBGCLLL 6.7 Ki 2
OSKBHMKTWRTXFP 6.7 Ki 2
PSMUPQQFBXUNIR 6.7 IC50 4
PUNXWODWMDLZDP 6.7 Ki 5
QCKCTTSCZBLBGX 6.7 Ki 3
RAVGDLZWTLVAPH 6.7 Ki 5
RRQQJDVDDCNRCT 6.7 Ki 2
SXWJLTLRDSROPE 6.7 Ki 2
UXDCCAQNEAFCIQ 6.7 IC50 4
VGSSLDYPUXVRJF 6.7 Ki 2
VHYUYQHTMPWAPK 6.7 Kd 5
ZCGQKZSNOODCBF 6.7 IC50 3
MJJALKDDGIKVBE 6.7 IC50 30 Yes
SIYLLGKDQZGJHK 6.7 IC50 13
BPJPUWVKKKMZBI 6.7 IC50 3
FJIIFJMUKPRFTH 6.7 Ki 2
HFBJHLOSPZYUBV 6.7 IC50 4
SSQJHXZOEJZLAK 6.7 Ki 4
CDDIWPZUHAJMSE 6.7 IC50 2
GCIWKIYFLXQBOA 6.7 IC50 2
LRBPZOOGQFAYKA 6.7 Kd 5
PNGMPCNVGUFXDA 6.7 IC50 2
FHJHJYBFXRHWSS 6.7 Ki 4
2D structure