Target Details
UniProt ACP11229
Gene SymbolCHRM1
Protein NameMuscarinic acetylcholine receptor M1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,571
  • Clinical molecules 35
  • Avg pChEMBL 7.27
Top Co-occurrence Targets
Active Molecules (1,571)
InChIKey pChEMBL Type Targets Clinical
VIOKBNDQBQFHDH 9.5 Kd 3
HILDNLJIJXAVHA 9.5 Ki 3
LZCOQTDXKCNBEE 9.5 Ki 5
FPCBWBHSQIVWBN 9.5 Ki 3
HLWLKLSVJQAUNS 9.5 Ki 3
YIMZVETVJULTMF 9.5 IC50 3
DFCLHAWGKPEFIX 9.5 Ki 5
GKNCQZVZUCNDGS 9.5 Ki 3
HGMITUYOCPPQLE 9.4 IC50 3
STCLPZTXPMXQOZ 9.4 Ki 3
DDAFFKQDEBQDHP 9.4 Ki 3
PMSLDIHTDBABLG 9.4 IC50 3
BDLKVZCRRROJRY 9.4 IC50 3
FJVQALKRJDSNIH 9.4 IC50 3
FWPIWVUMKDFZSR 9.4 IC50 3
JEEPGBSHIOBHQN 9.4 IC50 3
JZXJMFOSRNVGHQ 9.4 IC50 3
KMKLFKWYYAVHDZ 9.4 Ki 3
SWLGIXHESZQGPK 9.4 IC50 3
REMJCBLKEGJHMN 9.4 IC50 3
GPSZYYQYTBZUGG 9.4 IC50 3
MNHIAFLMHVAZPM 9.4 Ki 3
LIOWQNKZGLXNRL 9.4 IC50 3
RKUNBYITZUJHSG 9.4 Ki 5
XXWOCVWJOICKHA 9.3 Kd 5
OTOMMRFOLVUTLQ 9.3 Ki 3
KKEGQSSUXOGEAF 9.3 Ki 5
WCMVSMOIDILBOJ 9.3 Ki 5
LATYFBCANWEEBS 9.3 Ki 3
NDXFHBBFUCQHAL 9.3 Ki 5
OUUOAZNFNHOROT 9.3 Ki 3
UFSZYKLBZJNXLV 9.3 Ki 5
UVVAXSWZJPKXLR 9.2 Ki 3
BKJWZAJINPBJAC 9.2 Ki 2
ZPUIFOBXUIMYGP 9.2 IC50 3
QOXJSXPGWIRRNX 9.2 Ki 5
FLUDDWGSVPESJK 9.2 Ki 3
LAOBIJDCKIAALB 9.2 Kd 3
SPCFAZXKBQPYBW 9.2 Kd 3
ZMGKLIJUSAOHFP 9.2 IC50 3
KQCRPVVAJACIHG 9.2 Ki 3
VLCYSUDIOLZSJK 9.2 Ki 3
QCYOIEZHUQHFEJ 9.2 Ki 3
OLZRBZLJTKELRL 9.2 Ki 4
AVNRDCQRRUOTCC 9.2 Ki 5
GHHSRBSZNGGGPF 9.2 Ki 3
LVPIEYVPDBYBIT 9.1 Ki 3
PDEIQJDUHQRSQF 9.1 Ki 3
OYSTUJDZKCGRKD 9.1 Ki 3
UJXAGMVNACHDOG 9.1 Ki 5
2D structure