Target Details
UniProt ACP11229
Gene SymbolCHRM1
Protein NameMuscarinic acetylcholine receptor M1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,571
  • Clinical molecules 35
  • Avg pChEMBL 7.27
Top Co-occurrence Targets
Active Molecules (1,571)
InChIKey pChEMBL Type Targets Clinical
HCYAFALTSJYZDH 7.0 Ki 14 Yes
HXBKNTPSKWVIGR 7.0 Ki 4
KATNASIOTBDBDJ 7.0 IC50 2
MJUQLGDPJKYTLP 7.0 IC50 2
QSAKHCKHBZBOKB 7.0 IC50 4
ROJTXNMSUIEMFK 7.0 IC50 4
STUWFURQGSMWES 7.0 Ki 5
UAIKSDXRQZELHM 7.0 IC50 4
VUWOKTOQKPRPDM 7.0 Ki 5
WULCBOSTMCYKCZ 7.0 Kd 5
YTXILLIRPDSLHZ 7.0 Ki 5
ZZVUWRFHKOJYTH 7.0 Ki 11 Yes
BFELQLHLUNQIHL 7.0 Ki 5
QQPVAVCRPBYZDM 7.0 IC50 2
UXBPYISKBNGZMG 7.0 Ki 4
FPTVPLUMEFOZHQ 6.9 Ki 4
HJJPJSXJAXAIPN 6.9 IC50 3
QKTOQRPNKITPLN 6.9 IC50 5
RHAFROHARIZTPJ 6.9 Kd 5
BFELQLHLUNQIHL 6.9 Ki 2
REFOKOYWCWAHCW 6.9 IC50 3
VKQLNHVNHKXWJD 6.9 Ki 2
VPWKHNIBDCHPNN 6.9 Ki 5
AKLGENRCHBXEKW 6.9 Ki 3
AMKGONWYZZPTIL 6.9 IC50 4
DVVFXQIXRYZXNS 6.9 Ki 5
DYUCIPGRLQNPOD 6.9 IC50 4
FIMOHMGQXMTFNO 6.9 IC50 5
IJMVYQUDORUVOI 6.9 IC50 4
KHLGLAZJVORACT 6.9 Ki 3
KWBBYHOSQKDRRU 6.9 Ki 3
MHKMBBUFOBEBGG 6.9 IC50 2
NASFNLMUWVJIEY 6.9 Ki 5
ODRXKRITNIHJDG 6.9 IC50 4
RIJICWHWOASZHK 6.9 IC50 3
RIJICWHWOASZHK 6.9 IC50 3
UDXBARFJUKBPBJ 6.9 IC50 5
UUQSWYMJKUSTBX 6.9 Ki 5
VBPQNYMWBQALHS 6.9 Ki 5
VWBQUAMKHIBZSG 6.9 Ki 5
GGJSWQALDWFCMN 6.9 Ki 2
GKFAOGATDDYRDQ 6.9 Ki 5
RWZFXPOJQFVTQX 6.9 IC50 3
FHNLUXLINNMPIP 6.9 IC50 3
KQHKTHFVDIBYJZ 6.9 Ki 5
URKOMYMAXPYINW 6.9 Ki 27 Yes
YQUMEJDEWPVTIF 6.9 Kd 3
DSYOVHINHROBKN 6.9 IC50 4
DUEFVTWWBMZUOU 6.9 IC50 4
FVWZPHBNOSKYGM 6.9 IC50 4
2D structure