Target Details
UniProt ACP11229
Gene SymbolCHRM1
Protein NameMuscarinic acetylcholine receptor M1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,571
  • Clinical molecules 35
  • Avg pChEMBL 7.27
Top Co-occurrence Targets
Active Molecules (1,571)
InChIKey pChEMBL Type Targets Clinical
APULGHONBSGSEC 7.0 Ki 2
GNHXYBDOJNQUSM 7.0 Ki 4
PTBANFXYQIIDAF 7.0 Ki 5
XCSJIKDLUXGHQG 7.0 Ki 4
XKYMIJTXUGXDLR 7.0 Ki 4
YGBFXINLTZYAPY 7.0 Ki 2
DSPDJPFEBQTXDO 7.0 Kd 5
PQOOIERVZAXHBP 7.0 Ki 6
QCOZXCKWZLHYKC 7.0 Ki 4
AKPSMQSQINOOPH 7.0 Ki 5
BCPVTLUZROTVTR 7.0 IC50 4
BOAACWURMVXPFG 7.0 IC50 2
CYTRNWHHJCCGBY 7.0 IC50 4
DZIWUHCUDURPKK 7.0 IC50 3
FBYQQBWWVQINBI 7.0 IC50 4
GEALCDALCGCQFR 7.0 IC50 4
GHVVHNWTSPTZKS 7.0 IC50 4
GNEIWNURFQPOMA 7.0 IC50 3
GNHYCLNLNXMESJ 7.0 IC50 4
HYEGIQJKVHAAPE 7.0 IC50 2
ICAJLQZVLFKOOK 7.0 IC50 4
LCJWZLPNZLCYKB 7.0 Ki 5
PBCNZXLLSIAHHR 7.0 Ki 2
PULJCGFLKSMODH 7.0 Ki 4
QUYWXQCGHJOUSX 7.0 IC50 4
RJKOEXRPQFHGFU 7.0 IC50 4
RUCYNEILMKNPMV 7.0 IC50 4
UQSRLNYPAPLJBP 7.0 IC50 3
VAVAMZWIHKTIFJ 7.0 IC50 2
WGFZESGMAYFITP 7.0 IC50 4
WJIDIDMJHVMZSA 7.0 IC50 4
XYIJOTOXQIJOIN 7.0 Kd 5
XZPLJXKNDMOTKN 7.0 IC50 4
YYEWXNWXUYYCSF 7.0 IC50 3
AHOUBRCZNHFOSL 7.0 Ki 13
DUYRWEBTZNUILI 7.0 IC50 5
GTJOIOQFIDFYOI 7.0 Ki 4
PILDZUGYLLHLSW 7.0 IC50 2
WDLCZGMJXFWVAF 7.0 IC50 4
CKPSTQITKHNXIA 7.0 Ki 3
DPSJSZQSAMCEEQ 7.0 IC50 5
FMPNFDSPHNUFOS 7.0 Ki 5
FMPNFDSPHNUFOS 7.0 Ki 5
SXJIFPXBFXLADR 7.0 Ki 2
UWKMFEOQWPCWLU 7.0 Ki 5
AMKGONWYZZPTIL 7.0 IC50 4
BDHJGNMIOKDXBI 7.0 IC50 4
CITXQYRJEHWFPC 7.0 IC50 4
FUBPLGZZKBHUDG 7.0 IC50 4
FVXKERPIGVCGIR 7.0 IC50 4
2D structure