Target Details
UniProt ACP11229
Gene SymbolCHRM1
Protein NameMuscarinic acetylcholine receptor M1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,571
  • Clinical molecules 35
  • Avg pChEMBL 7.27
Top Co-occurrence Targets
Active Molecules (1,571)
InChIKey pChEMBL Type Targets Clinical
XJGVXQDUIWGIRW 7.2 Ki 17
ZTVIKZXZYLEVOL 7.2 IC50 5
HDACFKYOBJLCPQ 7.2 IC50 2
JOMFXRAREZYSMG 7.2 IC50 5
SVFAJETUQHWCFK 7.2 Ki 2
VQODXNCHOGDXSX 7.2 Ki 4
YZCWHHFUBMQIKE 7.2 Ki 5
ZQIYKYBVHCNJMX 7.2 IC50 5
AHQFYDVLGIPHDD 7.2 Ki 3
GGBGQOLEDWWRQA 7.2 Ki 2
HENUVGOJALLNNX 7.2 Ki 2
PYTIEHIIMNFIHE 7.2 Ki 3
RNNZREWYEVVFIS 7.2 IC50 4
SAPNXPWPAUFAJU 7.2 Ki 10
UUQSWYMJKUSTBX 7.2 Ki 5
DJIVSTFQGOLPFP 7.2 Ki 4
GTJOIOQFIDFYOI 7.2 Ki 4
IDIYVYIRDOLARV 7.2 IC50 4
KNYTYCPABXXTHV 7.2 Ki 3
LFWQLTRMYDLODO 7.2 IC50 4
RMIVAAULYORDDZ 7.2 Ki 2
TTYSIMLGCGISQV 7.2 IC50 4
UYTRDPRPLHVIIF 7.2 IC50 4
WGFZESGMAYFITP 7.2 IC50 4
WMPSFVBNWOMJKI 7.2 Ki 3
WXLHBKPIRLKYAH 7.2 IC50 5
XAPDCGAVGSRGKC 7.2 IC50 2
UPPZIKNLEDOKKO 7.2 Ki 5
NXIFJNOHOQFSCE 7.1 Ki 5
SEXKJERBKVAFLC 7.1 Ki 4
ZGVVXALTCVXMNS 7.1 Ki 2
KDMFWQZABCPNHX 7.1 Ki 2
KQJQPAOCEGFVNJ 7.1 IC50 3
WKEGMVFSZKEMJV 7.1 Ki 5
XELMJOZTBDQHDI 7.1 IC50 2
CFJMRBQWBDQYMK 7.1 Ki 4
GQAHLUHWIIZPFR 7.1 Ki 5
MXMXMYWNGBMDEJ 7.1 Ki 2
NCNQPLHOBSEBMQ 7.1 IC50 3
NSHSCDMDDQNBOD 7.1 Ki 2
XQNYYNJJJYBGLT 7.1 Ki 2
XUDSWTHYTNINGG 7.1 IC50 3
YPUMMBFUPIPODG 7.1 IC50 5
AESSYHBGSGYEPG 7.1 Ki 5
IVUOMTRDHAJWCR 7.1 IC50 4
KUKJOLRCPDCJAJ 7.1 Ki 5
MNTJDNKIZZJMSD 7.1 IC50 5
QTQLWKLZSPZQTO 7.1 Ki 5
QYBDNKCNIXORPK 7.1 Ki 2
CTFDKSWRIMHOOV 7.1 Kd 3
2D structure