Target Details
UniProt ACP11229
Gene SymbolCHRM1
Protein NameMuscarinic acetylcholine receptor M1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,571
  • Clinical molecules 35
  • Avg pChEMBL 7.27
Top Co-occurrence Targets
Active Molecules (1,571)
InChIKey pChEMBL Type Targets Clinical
SNSMIIQEKVYNOH 7.4 Ki 5
GTXZQPRWWKNJQL 7.4 Ki 5
IJRUGZIZSARHLR 7.4 Ki 5
UFUQREONAQKXQA 7.4 Ki 5
BFRFNKMZBSGKIG 7.3 Ki 3
FMMKJMIJNXFPMS 7.3 IC50 3
FNCJWKNHUAURLL 7.3 Ki 5
GDLIGKIOYRNHDA 7.3 IC50 24 Yes
PMCCMEISWXQOME 7.3 Kd 5
ZVNAONQCGLGOAO 7.3 Ki 3
GPFBOILGPPNQAT 7.3 Ki 4
YJWWBNSDIIFYRN 7.3 IC50 6 Yes
ZPEIMTDSQAKGNT 7.3 Ki 35 Yes
PIVCJDAJTNZQDR 7.3 Ki 3
AVNRDCQRRUOTCC 7.3 Ki 5
HNJAEIXPTNJDDI 7.3 Ki 5
QVYRGXJJSLMXQH 7.3 Ki 14
VSHUCQXNUSYTML 7.3 IC50 3
GMGHBSHBCGMTKY 7.3 IC50 3
PCVIRSOAUKEBJR 7.3 IC50 4
RWNXMLKAIWDHLU 7.3 IC50 5
UDXBARFJUKBPBJ 7.3 IC50 5
XCYNAFSXKQRKGO 7.3 Ki 5
YIDUXCASAXKJEC 7.3 Ki 5
ZUXRZVPVHVFNSX 7.3 IC50 5
FBOUYBDGKBSUES 7.3 Ki 6
ITDUNAGUAFBFRA 7.3 Ki 5
MIDPZKJBVKOKKF 7.3 Ki 3
CSHHMALNFJAJIB 7.3 Ki 2
FPDZLKMXESBTBK 7.3 Ki 3
MMHVHROUFYSFCY 7.3 Ki 3
MPVIJPUSNDEBBO 7.3 Ki 5
NFVADXLLOOOZIS 7.3 Ki 5
SWCMGAVLLBRPAS 7.3 Ki 3
APAQSJKHYTYKSS 7.3 IC50 3
CUCVCEWRTFMXDA 7.3 IC50 5
MTKHCEFATKQYMK 7.3 IC50 4
ZFXGEVATMHZGBZ 7.3 Ki 3
BZBLQCBDTFEROJ 7.3 Ki 3
HTYJHPPHBQRXGX 7.3 Ki 5
NQBTZXNQBCBXSM 7.3 Ki 3
PPZSYYWPALHGHI 7.3 Ki 2
RQJNIMUZOJATIT 7.3 Ki 3
RTNLSUYWOQRWMP 7.3 Ki 4
TWEXWSGNHKGNHI 7.3 Ki 4
UCDAGGLRRYYIRU 7.3 Ki 3
UEUYDRJDYJUBTN 7.3 Ki 3
WFHGMWHPBQUAFQ 7.3 Ki 3
WTNHCZORDQEROL 7.3 Ki 4
XELMJOZTBDQHDI 7.3 IC50 3
2D structure