Target Details
UniProt ACP11229
Gene SymbolCHRM1
Protein NameMuscarinic acetylcholine receptor M1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,571
  • Clinical molecules 35
  • Avg pChEMBL 7.27
Top Co-occurrence Targets
Active Molecules (1,571)
InChIKey pChEMBL Type Targets Clinical
FWARLZJUQIRKFD 7.5 Ki 3
MZDYABXXPZNUCT 7.5 Ki 5
RINSDLXTLQIMOU 7.5 Ki 4
BATVXAHTJHXAJQ 7.5 IC50 3
INAWHDCHKDVXJX 7.5 Ki 2
MXCOVFAJNYVLIQ 7.5 Kd 3
TWMXGXSGGIIQDM 7.5 Ki 5
OFBOKKRZVJJZHR 7.5 Ki 5
OUQAVICYOCWJLG 7.5 Ki 5
AHQFYDVLGIPHDD 7.5 Ki 3
AWOHFPFOFIIQDJ 7.5 IC50 3
FZOPOAUKSIMGRQ 7.5 Ki 2
UCHZYHUKFPSDLQ 7.5 IC50 3
ROCXJUPHBFOUQO 7.5 Ki 3
STXKNPNDRQOXKG 7.5 Ki 3
WCQIGWGZUOSGET 7.5 Ki 5
CPHUSFMAHLLFQS 7.5 IC50 5
DMQAXIJUTYJHIV 7.5 Ki 6
MDSAFGBQDVEKGD 7.5 IC50 3
YUCQRSFKFKVEJX 7.5 IC50 4
CHXGLJOIUDBPTI 7.5 Ki 5
OANBYDFPBWKVGI 7.5 Ki 5
BOXRBFJLKOMZNE 7.4 Ki 3
FFERIMSSXPDFOU 7.4 Ki 2
HXQMZFUQSGJNPQ 7.4 Ki 5
POGDAPYUQHRUOU 7.4 Ki 5
FRPQVLGDJMCCIJ 7.4 Ki 2
KWJMMMDBONQOQA 7.4 Ki 3
ODQWQRRAPPTVAG 7.4 IC50 20 Yes
WTWPGUIYLXNGRX 7.4 Ki 5
BCUGCHZRMKTPMU 7.4 Ki 6
GZCFTOXAOVPCDV 7.4 Ki 2
ODQWQRRAPPTVAG 7.4 Ki 14
UNZBDOQVZFAUNP 7.4 Ki 5
RTHXTYWCAPYZGF 7.4 Ki 3
YRIHWSWKYBUXOL 7.4 IC50 5
GSVREIJRMHEFJP 7.4 Kd 3
GVAQMKQFUDBPGS 7.4 IC50 3
HFMRXHYPEFDVMM 7.4 IC50 4
LDKQFEPUPKIHCG 7.4 Ki 2
NMLLDSGALUOMAS 7.4 IC50 3
NUTBZWNUSQLMQA 7.4 IC50 4
SNNFRAGGSGAUHH 7.4 IC50 3
UPDOKFNDDXFBCH 7.4 Ki 4
FNAJWFJEAUHFJC 7.4 Ki 2
GLRXSDVYMJTKAU 7.4 Ki 4
WQILUXNQRKEYJI 7.4 Ki 4
BCGWQEUPMDMJNV 7.4 Ki 30 Yes
FTFRVHRVNAJZCB 7.4 Ki 5
LNNRXCJKYSSUPF 7.4 Ki 3
2D structure