Target Details
UniProt ACP11229
Gene SymbolCHRM1
Protein NameMuscarinic acetylcholine receptor M1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,571
  • Clinical molecules 35
  • Avg pChEMBL 7.27
Top Co-occurrence Targets
Active Molecules (1,571)
InChIKey pChEMBL Type Targets Clinical
UWQNUCNXNKMWKG 7.7 Ki 5
UWVWASPAVBANND 7.7 Ki 5
VYVYCDJDMPVQTH 7.7 Ki 2
XMDRTFUFPOAGDR 7.7 Ki 9
YNNUSGIPVFPVBX 7.7 Ki 24 Yes
OTYJWRFICHGQJT 7.7 Ki 5
UKMOUADRKGHLMZ 7.7 Ki 3
UOKGNINOAYOIDX 7.7 Ki 5
VJJVBHULGOMODS 7.7 Ki 3
WXXOCGISBCTWPW 7.7 IC50 4
YRAPYXYTEMMURR 7.7 Ki 3
FNTHJTUPRVAXFZ 7.7 IC50 17
JIHUIMZDKDGEHR 7.7 Ki 2
KYYKFSMOYWOWFU 7.7 Ki 2
RHAFROHARIZTPJ 7.7 Kd 5
TWCQJLAORZMNFA 7.7 IC50 5
GPFBOILGPPNQAT 7.7 Ki 4
RVTKNIPUELNCNR 7.7 Ki 5
ARNGHJQKGZGVCU 7.6 Ki 2
GYWKQZUBLIAUNR 7.6 Ki 3
IABCBMLUYJFQMB 7.6 Ki 2
JNBDSWBJCGQGPV 7.6 Ki 5
MVNBPMNELMRFMU 7.6 Ki 5
NZWOPGCLSHLLPA 7.6 Ki 2
LPJZXUYTCJIHTG 7.6 Ki 5
PXFVYJJBXFKROG 7.6 Ki 3
GFDOCHMSKUCLIW 7.6 Ki 5
GRIVDARKNIXUML 7.6 IC50 3
RWNXMLKAIWDHLU 7.6 IC50 2
ZUXRZVPVHVFNSX 7.6 IC50 2
LMGYQTFTIFUZCP 7.6 IC50 2
PVJYTQKTDNFHQU 7.6 Ki 3
HRBJAGYSTCJZLI 7.6 Ki 2
IASYIMACMPYPDM 7.6 Ki 3
IXXCPZGOFVCPCH 7.6 Ki 5
QTBCATBNRIYMPB 7.6 Ki 5
XWGIZMOOTLOFBG 7.6 IC50 2
OJZRLJIPACRTSA 7.6 IC50 3
GZYGHLOFWVNJOI 7.5 IC50 3
KKSJQQXZULJWIM 7.5 Ki 2
KLQQZEIBZUZRLW 7.5 Ki 4
LOOAMMHLLVGAEL 7.5 Ki 5
LOZFSJRXJHXNTK 7.5 IC50 3
MGLYIVWWTWSJAF 7.5 IC50 4
UKIPQWNRWJEJMN 7.5 Ki 4
VGZCKWSRGATAFA 7.5 Ki 2
XSIRNWJXBZIYEQ 7.5 Ki 2
ZPMRLGPLMNVIDC 7.5 Ki 4
AYQKIBOBFAZBCX 7.5 Ki 5
CUYJUFFZSFIMQM 7.5 Ki 5
2D structure