Target Details
UniProt ACP11229
Gene SymbolCHRM1
Protein NameMuscarinic acetylcholine receptor M1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,571
  • Clinical molecules 35
  • Avg pChEMBL 7.27
Top Co-occurrence Targets
Active Molecules (1,571)
InChIKey pChEMBL Type Targets Clinical
LACTUOLELFMBLS 10.7 Ki 2
UKXSKSHDVLQNKG 10.4 Ki 5
IECFFSCULPEXHT 10.4 Kd 3
WNLPVNSWPNRWQU 10.4 Ki 2
BKLAJZNVMHLXAP 10.3 Ki 3
HGMITUYOCPPQLE 10.3 Ki 5
LERNTVKEWCAPOY 10.2 IC50 5
XXWOCVWJOICKHA 10.1 Kd 5
ASMXXROZKSBQIH 10.0 IC50 5
LERNTVKEWCAPOY 10.0 IC50 6
XQODGRWXBOXGGN 10.0 IC50 3
PRPBOUUIRMITJF 10.0 Ki 3
MTYMLJSBEPCLGC 9.9 IC50 3
WGOJWDWKHJHXSV 9.9 Ki 5
WCMVSMOIDILBOJ 9.9 Ki 5
CCXOXKSAHHQWSK 9.9 Ki 3
KBNPGVPUYYZVTB 9.9 Ki 3
NHUURXLCGOCXHZ 9.9 Ki 5
WOMCGBFNBSIIEA 9.9 Ki 5
ANGKOCUUWGHLCE 9.9 IC50 5
ROEXPZFFOZZHOY 9.9 Ki 5
FVTWTVQXNAJTQP 9.8 Ki 3
OLYUOAVKDLVFLJ 9.8 Ki 5
PMSLDIHTDBABLG 9.8 IC50 3
GWAMGWDJCYIREE 9.8 Kd 20
IWBMAAUPHUCYCI 9.8 Kd 20
MODBIBJHAWXYOZ 9.8 Kd 20
ZRQMUCDHVVOENY 9.8 Kd 17
RBDHPXXRYPWNOU 9.7 IC50 3
GYDFTKNRHZMENP 9.7 IC50 3
MYLRUMTYZFICQR 9.7 IC50 3
ZOZCBLGQKDOWFZ 9.7 Kd 3
MYLRUMTYZFICQR 9.6 IC50 3
NBQAKYWBUGUZTQ 9.6 IC50 3
VUHTYJDJRISPLZ 9.6 IC50 3
RBDHPXXRYPWNOU 9.6 IC50 3
WCMVSMOIDILBOJ 9.6 Ki 5
VJOYACFUOINUHV 9.6 IC50 3
GIJXKZJWITVLHI 9.6 IC50 16
GUWDPEQJYFKDCE 9.6 Ki 3
WOMCGBFNBSIIEA 9.6 Ki 5
QIEUGZFWENFVBK 9.6 IC50 3
RKUNBYITZUJHSG 9.5 Ki 5
TWCNWISPABVKII 9.5 IC50 3
ZYZIHJMWCSZLEQ 9.5 IC50 3
AFLBGAQHDSOPKA 9.5 Ki 5
UFSZYKLBZJNXLV 9.5 Ki 5
DAIWBMZPSVQRCH 9.5 IC50 3
NVEZMQGUUUDQFV 9.5 IC50 3
SIEQNGMENABBKP 9.5 Kd 3
2D structure