Target Details
| UniProt AC | P11166 |
|---|---|
| Gene Symbol | SLC2A1 |
| Protein Name | Solute carrier family 2, facilitated glucose transporter member 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00083 (Sugar_tr) |
Summary
- Multi-target molecules 189
- Clinical molecules 2
- Avg pChEMBL 7.11
KEGG Pathways (13)
- Adipocytokine signaling pathway
- Bile secretion
- Central carbon metabolism in cancer
- Diabetic cardiomyopathy
- Efferocytosis
- Glucagon signaling pathway
- HIF-1 signaling pathway
- Human T-cell leukemia virus 1 infection
- Insulin resistance
- Insulin secretion
- Pathways in cancer
- Renal cell carcinoma
- Thyroid hormone signaling pathway
Associated Diseases (5)
Active Molecules (189)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NFZSKIKFKFMYAP
|
6.8 | IC50 | 2 | — | |
ZFUNKFOMZPXBEZ
|
6.8 | IC50 | 2 | — | |
JMDDXCKPMOKCEA
|
6.8 | IC50 | 2 | — | |
VVWQJWNUSDWPGZ
|
6.8 | IC50 | 2 | — | |
HNFXFISXXNEMAC
|
6.8 | IC50 | 2 | — | |
BWJGMFCGWCHWCB
|
6.8 | IC50 | 2 | — | |
CCJSOPCDGNBPRQ
|
6.8 | IC50 | 2 | — | |
CIIAIZAOSYXJCJ
|
6.8 | IC50 | 2 | — | |
GVQCZFVGWQLYPD
|
6.8 | IC50 | 2 | — | |
HMDNBFHBMJGAQO
|
6.8 | IC50 | 2 | — | |
JQLUQQREDDBVIP
|
6.8 | IC50 | 2 | — | |
KOUVGGOMJZDBNK
|
6.8 | IC50 | 2 | — | |
NYOVTXRTDRFYKM
|
6.8 | IC50 | 2 | — | |
PGHDMVKHRCZCBN
|
6.8 | IC50 | 2 | — | |
VIPXMIJWKSZXNK
|
6.8 | IC50 | 2 | — | |
WHLMRVZMSUIARE
|
6.8 | IC50 | 2 | — | |
WTLQFUUVNBRDMG
|
6.8 | IC50 | 2 | — | |
YSRDLZNFOYOXDI
|
6.8 | IC50 | 2 | — | |
FEPKAPZLLAGREI
|
6.8 | IC50 | 3 | — | |
STAKKESPUWZRGP
|
6.7 | IC50 | 2 | — | |
WTNWZIWDNZGDTJ
|
6.7 | IC50 | 2 | — | |
HDMPSEDAIUYLPS
|
6.7 | IC50 | 3 | — | |
NRSNOIKPAFOCRX
|
6.7 | IC50 | 3 | — | |
QDGPJDFXLIQWGU
|
6.7 | IC50 | 3 | — | |
DENIPLMYQYHPPA
|
6.7 | IC50 | 6 | Yes | |
ZJQILEZGHUJAIA
|
6.7 | IC50 | 2 | — | |
KRJOUGBAJCNBKK
|
6.7 | IC50 | 3 | — | |
HXRCCVXGXJOFHE
|
6.6 | IC50 | 2 | — | |
ULOLUGXMKLIZGE
|
6.6 | IC50 | 8 | Yes | |
YPHMISFOHDHNIV
|
6.6 | IC50 | 6 | — | |
IXZVJTRRPOHKJF
|
6.6 | IC50 | 2 | — | |
TXYRCYTZTKAKKO
|
6.6 | Kd | 2 | — | |
WKLIILWHYTVQKO
|
6.6 | IC50 | 3 | — | |
AIRZCVGMOIZQHG
|
6.6 | IC50 | 2 | — | |
IUBIUOFPWZSBMU
|
6.6 | IC50 | 3 | — | |
AHOIVVKRHCTFHO
|
6.6 | IC50 | 2 | — | |
FYIWCUFRBHMEBW
|
6.6 | IC50 | 2 | — | |
MVDAZBJCOWDKRR
|
6.5 | IC50 | 3 | — | |
VWDJISBNSAISPO
|
6.5 | IC50 | 2 | — | |
VORLETARIHEPRV
|
6.5 | IC50 | 3 | — | |
NZDWQDUNLQVXSH
|
6.5 | IC50 | 2 | — | |
VFHBXTRXODMWII
|
6.5 | IC50 | 2 | — | |
YKJYKKNCCRKFSL
|
6.5 | IC50 | 3 | — | |
FYHUQCGSJPYQHW
|
6.5 | IC50 | 2 | — | |
AHCXENWSIKCTSI
|
6.5 | IC50 | 3 | — | |
JRQYXWVDIBVRHN
|
6.5 | IC50 | 3 | — | |
ZWFDKDJACHDCTD
|
6.5 | IC50 | 3 | — | |
BCJYPQKDTINZEK
|
6.4 | IC50 | 2 | — | |
BMUREBQUSAVLNX
|
6.4 | IC50 | 2 | — | |
BUVGDANTTMVYCT
|
6.4 | IC50 | 2 | — |