Target Details
| UniProt AC | P11166 |
|---|---|
| Gene Symbol | SLC2A1 |
| Protein Name | Solute carrier family 2, facilitated glucose transporter member 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00083 (Sugar_tr) |
Summary
- Multi-target molecules 189
- Clinical molecules 2
- Avg pChEMBL 7.11
KEGG Pathways (13)
- Adipocytokine signaling pathway
- Bile secretion
- Central carbon metabolism in cancer
- Diabetic cardiomyopathy
- Efferocytosis
- Glucagon signaling pathway
- HIF-1 signaling pathway
- Human T-cell leukemia virus 1 infection
- Insulin resistance
- Insulin secretion
- Pathways in cancer
- Renal cell carcinoma
- Thyroid hormone signaling pathway
Associated Diseases (5)
Active Molecules (189)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QJMMARYXYAZEQD
|
9.5 | IC50 | 3 | — | |
CJLYRRJNZDMNNV
|
9.0 | IC50 | 3 | — | |
JPBASMDABOPXNH
|
9.0 | IC50 | 2 | — | |
NLIRYBSWIKFCMB
|
9.0 | IC50 | 3 | — | |
UELMPNTWJSQIOB
|
9.0 | IC50 | 2 | — | |
FVCHETZUBCPYNZ
|
8.7 | IC50 | 2 | — | |
HWBKGCWYDNMKRS
|
8.5 | IC50 | 3 | — | |
LGMLKXQXZUDVPY
|
8.5 | IC50 | 3 | — | |
MDTIVUPPYRUWIP
|
8.5 | IC50 | 2 | — | |
PQXLHNMQCBOGJS
|
8.5 | IC50 | 3 | — | |
CJDVUGHFAUGCOI
|
8.4 | IC50 | 2 | — | |
NCPQJZBOWARLET
|
8.4 | IC50 | 2 | — | |
UBPDZSOJWGTGPP
|
8.4 | IC50 | 3 | — | |
FDPVPDHJOTXXCZ
|
8.3 | IC50 | 3 | — | |
HBXKXXRRQJIJRG
|
8.3 | IC50 | 3 | — | |
LHQZZJAIOHNXKA
|
8.3 | IC50 | 2 | — | |
QPRAMIWFCPMHCD
|
8.3 | IC50 | 2 | — | |
WGNKZDNKYFHWCC
|
8.3 | IC50 | 3 | — | |
HYYHSHCGRMCRCS
|
8.2 | IC50 | 2 | — | |
OHKDHHSQSZVIMW
|
8.2 | IC50 | 3 | — | |
BIEISOHNYWNUIA
|
8.2 | IC50 | 2 | — | |
DXJIXNIYGMNIFL
|
8.2 | IC50 | 2 | — | |
GDJUIVIIRPZSJR
|
8.2 | IC50 | 3 | — | |
UQYWHYXGIIUVRF
|
8.2 | IC50 | 3 | — | |
WEPMLRNQXNAKDE
|
8.2 | IC50 | 2 | — | |
HJZKOBOALSFQEU
|
8.1 | IC50 | 2 | — | |
OKRVHKNCIFLKMU
|
8.1 | IC50 | 2 | — | |
OSHZPHMMCGCAMN
|
8.1 | IC50 | 2 | — | |
JFCBFXVYBVDLSU
|
8.1 | IC50 | 3 | — | |
SJHQCCAIPHHSPI
|
8.1 | IC50 | 2 | — | |
CWASUJBNRKHFHU
|
8.0 | IC50 | 2 | — | |
UBSRKRDOZPXAES
|
8.0 | IC50 | 2 | — | |
WCYMZGBRFVGEJB
|
8.0 | IC50 | 3 | — | |
PMJSQDNDKVLTDZ
|
8.0 | IC50 | 2 | — | |
PBKOSJBDJUDWRP
|
7.9 | IC50 | 2 | — | |
MTIZOXXUAPPZTG
|
7.8 | IC50 | 2 | — | |
UGXJUOXVOVKIPG
|
7.8 | IC50 | 2 | — | |
DBMPNCBTGSGUJB
|
7.8 | IC50 | 2 | — | |
ONEQVTDJEHHOEX
|
7.8 | IC50 | 2 | — | |
BSLRZBMEFPHGBR
|
7.8 | IC50 | 3 | — | |
LUHHNRVUIPBDCT
|
7.7 | IC50 | 2 | — | |
MZXGHIXHMAWJJF
|
7.7 | IC50 | 2 | — | |
BKLJDIJJOOQUFG
|
7.6 | IC50 | 2 | — | |
DWZIDNSMNVRATG
|
7.6 | IC50 | 2 | — | |
JFBXEXDZHRGQKW
|
7.6 | IC50 | 2 | — | |
YAJBHJCFOICLGO
|
7.6 | IC50 | 2 | — | |
SPRLNKQKOJIGIN
|
7.5 | IC50 | 3 | — | |
SLJHJMKUVDGUKD
|
7.5 | IC50 | 2 | — | |
JSCZYXYOGWTKPQ
|
7.5 | IC50 | 2 | — | |
OBLZUEWTOIEOKI
|
7.5 | IC50 | 2 | — |