Target Details
| UniProt AC | P11137 |
|---|---|
| Gene Symbol | MAP2 |
| Protein Name | Microtubule-associated protein 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08377 (MAP2_projctn) PF00418 (Tubulin-binding) |
Summary
- Multi-target molecules 52
- Clinical molecules 0
- Avg pChEMBL 7.43
KEGG Pathways (1)
Active Molecules (52)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SCPCVOHBNFGSEL
|
8.5 | IC50 | 3 | — | |
KVBBKLNPTAGDQO
|
8.4 | IC50 | 2 | — | |
NIDNKFIXOVDXKL
|
8.4 | IC50 | 3 | — | |
BGVWCIRYUNODHW
|
8.3 | IC50 | 2 | — | |
BNTAEJNPQLMGDJ
|
8.3 | IC50 | 2 | — | |
LJBIQXKUSNRCSD
|
8.3 | IC50 | 3 | — | |
LMOBUEBHMONFLE
|
8.3 | IC50 | 3 | — | |
PWRMQUDNGXLDFA
|
8.3 | IC50 | 2 | — | |
PWRMQUDNGXLDFA
|
8.3 | IC50 | 2 | — | |
BNTAEJNPQLMGDJ
|
8.2 | IC50 | 2 | — | |
WBTSXAUWFXDAGS
|
8.2 | IC50 | 3 | — | |
OTERKSQZXOAQLU
|
8.2 | IC50 | 2 | — | |
RZXSROGFHJQWNH
|
8.2 | IC50 | 2 | — | |
MSIBXQCGLUUGLM
|
8.1 | IC50 | 3 | — | |
NLPCFFYBCGCRIT
|
8.1 | IC50 | 2 | — | |
OXGYZBBLOABNDR
|
8.1 | IC50 | 3 | — | |
PEWYGTLRHLRPDV
|
8.1 | IC50 | 3 | — | |
PYSBUBPDECGJSZ
|
8.1 | IC50 | 3 | — | |
VJZBRXPAQJXJPH
|
8.1 | IC50 | 3 | — | |
AUHZWZZQQBRYMA
|
8.0 | IC50 | 3 | — | |
IUZBXISRROMZSL
|
8.0 | IC50 | 2 | — | |
RRCNPYRCOUOTDZ
|
8.0 | IC50 | 2 | — | |
SERKGWYXQDCJCM
|
8.0 | IC50 | 2 | — | |
ZXWANJABEMQGRP
|
8.0 | IC50 | 2 | — | |
BPCCTTNRJCTGHS
|
7.9 | IC50 | 3 | — | |
MQBAPASGXUTVKD
|
7.9 | IC50 | 2 | — | |
BHMRWHRWBMLFNH
|
7.8 | IC50 | 2 | — | |
ORZCBQVVROFUNM
|
7.7 | IC50 | 2 | — | |
ZIWPWJYKIWRJHS
|
7.7 | IC50 | 2 | — | |
WNDUVATWTRICIS
|
7.4 | IC50 | 2 | — | |
PFAFARJWFBPNIN
|
7.3 | IC50 | 2 | — | |
VVDKBODANWRILU
|
7.2 | IC50 | 2 | — | |
IIJFTAYSJAHBBL
|
7.1 | IC50 | 2 | — | |
QHDWHCBIHPDKKB
|
7.1 | IC50 | 2 | — | |
ATBRTSOQFVTTON
|
7.0 | IC50 | 2 | — | |
BCTCNJXSYRAZDU
|
7.0 | IC50 | 2 | — | |
AKSQBPCRIODOMP
|
6.9 | IC50 | 2 | — | |
OXGKPVIBOVJKSI
|
6.7 | IC50 | 2 | — | |
FTRFOFPAMKYZPH
|
6.6 | IC50 | 4 | — | |
QPVQIYYFNNDMOE
|
6.6 | IC50 | 2 | — | |
NAOYSRBUEYWQNL
|
6.5 | IC50 | 3 | — | |
WSQQTUKKGLYHCD
|
6.4 | IC50 | 2 | — | |
DUYDXTWDEKJZHW
|
6.3 | IC50 | 2 | — | |
KEKIZDKQHXXAEP
|
6.3 | IC50 | 2 | — | |
KZDTUSZNJHGAIW
|
6.2 | IC50 | 2 | — | |
SXTKECRQJMUZOI
|
6.2 | IC50 | 2 | — | |
YYZBXLHPDIWNHC
|
6.1 | IC50 | 2 | — | |
JYZRJSXLGQYLJB
|
6.0 | IC50 | 2 | — | |
JTJRNFGGGCLXSL
|
6.0 | IC50 | 2 | — | |
PKAMRWQMJQIISK
|
6.0 | IC50 | 2 | — |