Target Details
| UniProt AC | P10828 |
|---|---|
| Gene Symbol | THRB |
| Protein Name | Thyroid hormone receptor beta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 210
- Clinical molecules 0
- Avg pChEMBL 8.04
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (210)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DSBHFVFSZGOWJG
|
7.3 | Kd | 2 | — | |
HFNOBCLNQQFRAY
|
7.3 | Kd | 2 | — | |
DXDHCVCAJKZAHT
|
7.3 | IC50 | 2 | — | |
DYNDGIZYGFNWSL
|
7.3 | Ki | 2 | — | |
LOFMSGBJMJLFHW
|
7.3 | Kd | 2 | — | |
YCQCSJYPJDNFIL
|
7.3 | Kd | 2 | — | |
QOWDVYZPDZEOEA
|
7.3 | IC50 | 2 | — | |
TWYFELLCKHAKCY
|
7.3 | IC50 | 2 | — | |
XSRIPYSSPXVKKY
|
7.3 | Ki | 2 | — | |
HZKLLZGFRIQXJL
|
7.2 | IC50 | 2 | — | |
LKIKBJBECFALSP
|
7.2 | IC50 | 2 | — | |
CMUXOLOARGWVNN
|
7.2 | IC50 | 2 | — | |
LGLKAFDDFXJFCK
|
7.2 | Kd | 2 | — | |
LLTQMRYGMABCOB
|
7.2 | Kd | 2 | — | |
UGVNVZOKSDTCKR
|
7.2 | IC50 | 2 | — | |
WGALZWWKJHCIBC
|
7.2 | IC50 | 3 | — | |
CQFMEEGANZACLR
|
7.1 | IC50 | 3 | — | |
DBSWHCJBBYJIJU
|
7.1 | IC50 | 2 | — | |
GZPZKAZISNKHLE
|
7.1 | Ki | 2 | — | |
KVHGFYBGJGPWIL
|
7.1 | IC50 | 2 | — | |
SGMXHEIWJQTVMJ
|
7.1 | IC50 | 3 | — | |
AWOYKHJWMXPCTQ
|
7.0 | Kd | 2 | — | |
OYZZBRHSILKBDZ
|
7.0 | Ki | 2 | — | |
RGPPXBMUCFRACH
|
7.0 | Kd | 2 | — | |
AOTADNCHLKUEAX
|
7.0 | IC50 | 2 | — | |
CXFUMQXKEITWKR
|
7.0 | IC50 | 2 | — | |
OSDJZABHEFWQAU
|
6.9 | IC50 | 2 | — | |
XWCKALNSQFREFM
|
6.9 | Kd | 2 | — | |
ZBRXDMONGVUIEW
|
6.9 | Kd | 2 | — | |
PUUWWSIUTRYHMF
|
6.9 | IC50 | 2 | — | |
VURXPVGLFFQSLT
|
6.8 | Kd | 2 | — | |
IKJMJDPMGHFSNH
|
6.8 | IC50 | 2 | — | |
NNEWESUWHJGSMJ
|
6.8 | IC50 | 2 | — | |
ANMSUCKVCVQUCL
|
6.7 | IC50 | 2 | — | |
LWSPPCNYLDHZNN
|
6.7 | IC50 | 2 | — | |
UQABRPIJAIHKQN
|
6.7 | IC50 | 2 | — | |
UUPVEFMYALNSEQ
|
6.7 | IC50 | 2 | — | |
ZCVQDNGOBFARHQ
|
6.6 | IC50 | 2 | — | |
BPCRJQJRJFLQHV
|
6.6 | Ki | 2 | — | |
NCPFGULZSPSFGH
|
6.6 | IC50 | 2 | — | |
ZZFTXXUUQNBOGX
|
6.5 | Kd | 2 | — | |
PVUIJHOHMVLYQT
|
6.5 | IC50 | 2 | — | |
GZEXEJKRKKWNSD
|
6.5 | Ki | 2 | — | |
ADOIUCPAWXGJSR
|
6.5 | IC50 | 2 | — | |
JQLXLCYSWMVCLC
|
6.5 | IC50 | 2 | — | |
FVDRTJXVCUAOCA
|
6.4 | IC50 | 2 | — | |
RPFZTCWLIDXIQK
|
6.4 | IC50 | 2 | — | |
LCTMPMFLXABADB
|
6.3 | IC50 | 2 | — | |
CJHLRGCXPGIPCB
|
6.2 | Kd | 2 | — | |
BSXKQZASVPAQPC
|
6.2 | IC50 | 2 | — |