Target Details
| UniProt AC | P10827 |
|---|---|
| Gene Symbol | THRA |
| Protein Name | Thyroid hormone receptor alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 194
- Clinical molecules 1
- Avg pChEMBL 7.32
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (194)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DYNDGIZYGFNWSL
|
6.5 | Ki | 2 | — | |
GZEXEJKRKKWNSD
|
6.5 | Ki | 2 | — | |
ZOOUPJHRNKSBCT
|
6.5 | IC50 | 2 | — | |
RGPPXBMUCFRACH
|
6.5 | Kd | 2 | — | |
LDAQJAHGYVAIQJ
|
6.5 | IC50 | 2 | — | |
OSDJZABHEFWQAU
|
6.4 | IC50 | 2 | — | |
NNEWESUWHJGSMJ
|
6.4 | IC50 | 2 | — | |
HAUMMAHCGKEHHL
|
6.4 | Ki | 2 | — | |
BNBWGVDBRHRJFJ
|
6.4 | IC50 | 2 | — | |
AWOYKHJWMXPCTQ
|
6.4 | Kd | 2 | — | |
JKQNTBZKAUPEAD
|
6.4 | Ki | 2 | — | |
QEDNCYVOSFGOAX
|
6.4 | IC50 | 2 | — | |
ANMSUCKVCVQUCL
|
6.3 | IC50 | 2 | — | |
AQOFZDMQOFEIFY
|
6.3 | IC50 | 2 | — | |
PVUIJHOHMVLYQT
|
6.3 | IC50 | 2 | — | |
UQABRPIJAIHKQN
|
6.3 | IC50 | 2 | — | |
UUPVEFMYALNSEQ
|
6.3 | IC50 | 2 | — | |
KVHGFYBGJGPWIL
|
6.3 | IC50 | 2 | — | |
NSMJTCRIXMAXDP
|
6.3 | Kd | 2 | — | |
HZKLLZGFRIQXJL
|
6.3 | IC50 | 2 | — | |
LWSPPCNYLDHZNN
|
6.3 | IC50 | 2 | — | |
NPKNCAXKMZYAIJ
|
6.3 | Ki | 2 | — | |
UGVNVZOKSDTCKR
|
6.3 | IC50 | 2 | — | |
WCRWBJJFDPTIQX
|
6.3 | IC50 | 2 | — | |
AGCPOGPDHHGRRI
|
6.2 | IC50 | 2 | — | |
GZPZKAZISNKHLE
|
6.2 | Ki | 2 | — | |
BSXKQZASVPAQPC
|
6.2 | IC50 | 2 | — | |
FVDRTJXVCUAOCA
|
6.2 | IC50 | 2 | — | |
RPFZTCWLIDXIQK
|
6.2 | IC50 | 2 | — | |
NCPFGULZSPSFGH
|
6.2 | IC50 | 2 | — | |
YFEVUUNMUSDKFZ
|
6.2 | IC50 | 2 | — | |
HHSRCUBLBZYJPA
|
6.2 | IC50 | 2 | — | |
IYIKLHRQXLHMJQ
|
6.2 | IC50 | 18 | — | |
ZIRMTIREZHSURE
|
6.2 | IC50 | 2 | — | |
ZCVQDNGOBFARHQ
|
6.2 | IC50 | 2 | — | |
VJKVJESSSPWLJY
|
6.2 | IC50 | 2 | — | |
XSRIPYSSPXVKKY
|
6.2 | Ki | 2 | — | |
ZDCMJDVSSLHLLQ
|
6.1 | Ki | 9 | Yes | |
BQVSQVFXKGWCRD
|
6.1 | IC50 | 2 | — | |
INJFUZZLERLMQZ
|
6.1 | Ki | 2 | — | |
LCTMPMFLXABADB
|
6.1 | IC50 | 2 | — | |
WDJZIEHFYCTEMU
|
6.1 | IC50 | 2 | — | |
DBSWHCJBBYJIJU
|
6.1 | IC50 | 2 | — | |
OYZZBRHSILKBDZ
|
6.0 | Ki | 2 | — |