Target Details
| UniProt AC | P10827 |
|---|---|
| Gene Symbol | THRA |
| Protein Name | Thyroid hormone receptor alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 194
- Clinical molecules 1
- Avg pChEMBL 7.32
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (194)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IXMROOKFPWGDGF
|
7.0 | IC50 | 2 | — | |
LZJNSIDSVOXSRG
|
7.0 | IC50 | 2 | — | |
COOBJKRJONOFHD
|
7.0 | IC50 | 2 | — | |
LKIKBJBECFALSP
|
7.0 | IC50 | 2 | — | |
SUEICZCJKXGOAJ
|
7.0 | IC50 | 2 | — | |
URFQJEGLROMZOX
|
7.0 | IC50 | 2 | — | |
AVSKLCKLTAIMHU
|
7.0 | IC50 | 2 | — | |
VURXPVGLFFQSLT
|
7.0 | Kd | 2 | — | |
JDRBJNQCUWNMPX
|
6.9 | IC50 | 2 | — | |
NHYQPCDQZSMCBN
|
6.9 | IC50 | 2 | — | |
BWPGMDHCTINHBA
|
6.9 | Ki | 2 | — | |
DBQMSDVEQUDKDW
|
6.9 | IC50 | 2 | — | |
JWLVVPFLXSEKNK
|
6.9 | IC50 | 2 | — | |
VQOQTSKXKNWJJY
|
6.9 | Ki | 2 | — | |
YTJRUGBPZHFBMK
|
6.9 | IC50 | 2 | — | |
SQDDKKYHCKRAHR
|
6.9 | IC50 | 2 | — | |
TVQYCFFCYRSFQF
|
6.9 | IC50 | 2 | — | |
PUUWWSIUTRYHMF
|
6.8 | IC50 | 2 | — | |
YYSMKKABVHWWAR
|
6.8 | Ki | 2 | — | |
MEAGUOMGJAPVGX
|
6.8 | Ki | 2 | — | |
OBCTYXFEJVMWDM
|
6.8 | Ki | 2 | — | |
PVUIJHOHMVLYQT
|
6.8 | IC50 | 2 | — | |
FWJUTJOHYIEPMV
|
6.8 | IC50 | 2 | — | |
DJHXUFXPDYXOPH
|
6.8 | Ki | 2 | — | |
NHIDWXMLJGPDMM
|
6.7 | Ki | 2 | — | |
VBUJXSSBBJJPKZ
|
6.7 | Ki | 2 | — | |
WTEXNXXPHWVVDS
|
6.7 | Ki | 2 | — | |
ADOIUCPAWXGJSR
|
6.7 | IC50 | 2 | — | |
QOWDVYZPDZEOEA
|
6.7 | IC50 | 2 | — | |
RKNMDWYQIVLKAB
|
6.7 | Ki | 2 | — | |
LDLCVNDDYJKRGP
|
6.7 | Ki | 2 | — | |
NDQVMFFAGUMNGI
|
6.7 | Ki | 2 | — | |
PBZAEAFSLYJVGD
|
6.7 | Kd | 2 | — | |
QFHPGLKTTMRBBJ
|
6.7 | IC50 | 2 | — | |
XYJAEXLTNMFZDJ
|
6.7 | IC50 | 2 | — | |
DIKMHXCTJKLLMY
|
6.6 | IC50 | 2 | — | |
NUVOUOHXOKZTQW
|
6.6 | IC50 | 2 | — | |
XGBAZMQYQFUGHW
|
6.6 | Ki | 2 | — | |
OKARMSOGGGWFDN
|
6.6 | Ki | 2 | — | |
DFUILVXTAGCSOH
|
6.6 | IC50 | 2 | — | |
HGCHTOCFDDIWOI
|
6.6 | Kd | 2 | — | |
MXHYBOCRTUHWOD
|
6.6 | IC50 | 2 | — | |
YFRJTYUEWKCLLN
|
6.6 | IC50 | 2 | — | |
DXDHCVCAJKZAHT
|
6.6 | IC50 | 2 | — | |
UTTJYFMWZBKOLA
|
6.6 | IC50 | 2 | — | |
CMUXOLOARGWVNN
|
6.6 | IC50 | 2 | — | |
IIYKWHVHNIUBER
|
6.5 | IC50 | 2 | — | |
AKEHDUZHUGHYIV
|
6.5 | Ki | 2 | — | |
ZZFTXXUUQNBOGX
|
6.5 | Kd | 2 | — | |
GHFDFTOECTVGNW
|
6.5 | IC50 | 2 | — |