Target Details
| UniProt AC | P10721 |
|---|---|
| Gene Symbol | KIT |
| Protein Name | Mast/stem cell growth factor receptor Kit |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,134
- Clinical molecules 305
- Avg pChEMBL 7.36
KEGG Pathways (11)
Associated Diseases (7)
Active Molecules (1,134)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BTDHMLNFQMGPGD
|
7.7 | IC50 | 3 | Yes | |
BYQDPWAYLMNNKF
|
7.7 | IC50 | 5 | Yes | |
DIEURDLEWWOVNF
|
7.7 | IC50 | 2 | — | |
IQOAIXAFDYRGNK
|
7.7 | IC50 | 3 | — | |
KVBWCMRDDFWCKD
|
7.7 | IC50 | 2 | — | |
QJSDPLBJLHJTJP
|
7.7 | IC50 | 6 | — | |
YTHUQGIGAIZNIM
|
7.7 | IC50 | 3 | — | |
FLYZOVOQWUDRBN
|
7.6 | IC50 | 2 | Yes | |
IFFBOVLYGJAFKB
|
7.6 | IC50 | 5 | — | |
PUPCRRRSBUYJAD
|
7.6 | IC50 | 44 | Yes | |
PZINVJUNZRLUIM
|
7.6 | IC50 | 3 | — | |
XOOCFOXUQTWFFJ
|
7.6 | IC50 | 5 | Yes | |
BHSOPYVVEZFHDB
|
7.6 | IC50 | 25 | Yes | |
DJRIFOSSHAVNOW
|
7.6 | IC50 | 2 | — | |
DNQBBKLYBVCDBY
|
7.6 | IC50 | 2 | — | |
FFJSXPWNHROKBN
|
7.6 | IC50 | 2 | — | |
MLFZJIDNGFABRH
|
7.6 | IC50 | 3 | — | |
GALVWTFFXPRMQM
|
7.6 | Ki | 20 | — | |
GXFMUXGPPXGMTM
|
7.6 | IC50 | 2 | Yes | |
LQXIQYJEMNHPCH
|
7.6 | IC50 | 2 | Yes | |
NRGYZNJPCGRCLV
|
7.6 | Ki | 52 | — | |
OWFXKTOLFUQPDJ
|
7.6 | Ki | 36 | — | |
SLZDAHQKZCFNCA
|
7.6 | IC50 | 3 | — | |
XJSFDMGICAWQFS
|
7.6 | Ki | 60 | — | |
YNVQXAFBFLYMLM
|
7.6 | IC50 | 3 | Yes | |
YZNNUIOSLHHWJF
|
7.6 | IC50 | 2 | Yes | |
HWEBFAZCYKVEJD
|
7.6 | IC50 | 5 | — | |
QFPRMYTURWHCEE
|
7.6 | IC50 | 3 | Yes | |
UXXQOJXBIDBUAC
|
7.6 | Kd | 21 | Yes | |
CQQHPXAPMGAALV
|
7.6 | IC50 | 4 | Yes | |
JPKSISIJPSXDLA
|
7.6 | IC50 | 10 | Yes | |
JVGNHFZOVWJKER
|
7.6 | IC50 | 3 | — | |
MDWDLNIDUNDEFN
|
7.6 | IC50 | 2 | — | |
QPSVRPUGGFUWCH
|
7.6 | IC50 | 2 | — | |
ATULXEYLXXNOLJ
|
7.6 | IC50 | 3 | — | |
DIOLCKJIPOAFOB
|
7.6 | IC50 | 2 | Yes | |
GJYHDNFJPKFHRH
|
7.6 | Ki | 4 | Yes | |
GWOSGFTZTVFDGQ
|
7.6 | IC50 | 5 | Yes | |
JGWRKYUXBBNENE
|
7.6 | IC50 | 11 | — | |
KNKIKEKAVNITNK
|
7.6 | IC50 | 3 | Yes | |
KWHMNEURGOHDLA
|
7.6 | IC50 | 2 | — | |
KXHOCICVTKWLSA
|
7.6 | Ki | 3 | — | |
ROYLPDZGPLFQSV
|
7.6 | IC50 | 3 | — | |
TVECXYJHKWEHKM
|
7.6 | IC50 | 2 | — | |
VKBFHTIUXUCYRQ
|
7.6 | IC50 | 8 | — | |
AHORVICCHQDIIL
|
7.6 | IC50 | 2 | — | |
ANKWXLPVGDMRLF
|
7.6 | Ki | 2 | — | |
AVRDADHHFBZKMF
|
7.6 | Ki | 2 | — | |
AYOKLOOUEVPQDU
|
7.6 | Ki | 2 | — | |
BKAAWAAYNIFIHU
|
7.6 | Ki | 2 | — |