Target Details
| UniProt AC | P10721 |
|---|---|
| Gene Symbol | KIT |
| Protein Name | Mast/stem cell growth factor receptor Kit |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,134
- Clinical molecules 305
- Avg pChEMBL 7.36
KEGG Pathways (11)
Associated Diseases (7)
Active Molecules (1,134)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VJRMARZDCXLFER
|
7.8 | IC50 | 3 | — | |
XOSIKVLXVWWHON
|
7.8 | IC50 | 3 | — | |
YBPBYWHVRLZISQ
|
7.8 | IC50 | 3 | — | |
ZVVIKPIHXSNXJY
|
7.8 | IC50 | 4 | Yes | |
HQVKWOAGEPGZAS
|
7.8 | IC50 | 3 | Yes | |
ODPGGGTTYSGTGO
|
7.8 | Kd | 153 | — | |
KIXJPVWFCZCXOL
|
7.7 | IC50 | 4 | Yes | |
RAKQGQRMHIXLRO
|
7.7 | IC50 | 3 | — | |
SFNDRKNZETUTKF
|
7.7 | IC50 | 5 | Yes | |
UKSRSPVTFVLKRY
|
7.7 | IC50 | 4 | Yes | |
XTMWIEVQVYQIFB
|
7.7 | IC50 | 2 | Yes | |
ZXQPAYCROYPEFR
|
7.7 | IC50 | 4 | Yes | |
BLXZMOITRCHHRV
|
7.7 | IC50 | 2 | Yes | |
DKDIYRYSJHNWTO
|
7.7 | IC50 | 2 | Yes | |
FTTJIZHHPOGNQH
|
7.7 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
7.7 | Kd | 408 | — | |
HKSZLNNOFSGOKW
|
7.7 | Kd | 49 | Yes | |
JUPMOGJCVRJIHK
|
7.7 | IC50 | 3 | Yes | |
KVDZJYLUBBYJIX
|
7.7 | IC50 | 2 | — | |
NWAUBAGBGOPJLF
|
7.7 | IC50 | 51 | Yes | |
QDCNUYNTRDKBDB
|
7.7 | IC50 | 3 | — | |
RPRCCKYNDFQWHV
|
7.7 | IC50 | 3 | — | |
ZPVUIOVIUFJGHO
|
7.7 | IC50 | 2 | — | |
NMGPNPSPONCMOZ
|
7.7 | IC50 | 3 | — | |
UHEXEECCTNTZTE
|
7.7 | Ki | 3 | — | |
WPHKIQPVPYJNAX
|
7.7 | IC50 | 81 | — | |
AAVMTXYKUJWQBU
|
7.7 | IC50 | 8 | Yes | |
ADLODFKELCDENP
|
7.7 | IC50 | 3 | — | |
BNVPFDRNGHMRJS
|
7.7 | IC50 | 3 | — | |
CFDOBTIFMPKBRD
|
7.7 | IC50 | 2 | — | |
HXUZQEYFKAZBPX
|
7.7 | IC50 | 4 | Yes | |
KLHJDCUHOKZNOP
|
7.7 | IC50 | 5 | Yes | |
LDACHLNBCOVNBL
|
7.7 | IC50 | 8 | — | |
MJDGTEDIUFSUBR
|
7.7 | IC50 | 2 | — | |
MQRDVGBWWVWMEN
|
7.7 | Ki | 47 | — | |
NRCYJQOXMJLQTP
|
7.7 | IC50 | 2 | Yes | |
QBRQTJMZEYORSP
|
7.7 | IC50 | 12 | — | |
QJJXDLUIDBRYRG
|
7.7 | IC50 | 3 | — | |
RPCMGDNNIFRGGQ
|
7.7 | IC50 | 4 | Yes | |
SCUGTCMSRMQNNQ
|
7.7 | IC50 | 7 | — | |
UKYJKXMPIDEQFF
|
7.7 | IC50 | 16 | — | |
UTQPKPHUIMHAAN
|
7.7 | Ki | 22 | — | |
UGVHUUTVPLIEGT
|
7.7 | IC50 | 2 | — | |
MHITTXFPZXWLMH
|
7.7 | Kd | 6 | — | |
PSNOTDXLJIXMTC
|
7.7 | IC50 | 4 | Yes | |
TZOUNCJSFSDDCR
|
7.7 | IC50 | 5 | Yes | |
UYWCBKUMESQOKL
|
7.7 | IC50 | 5 | — | |
WCDZEMSHEVLSFK
|
7.7 | Ki | 3 | Yes | |
JFYAFMMSOVKSEU
|
7.7 | IC50 | 4 | — | |
VSVJBCKLXDHEJV
|
7.7 | IC50 | 6 | — |