Target Details
| UniProt AC | P10721 |
|---|---|
| Gene Symbol | KIT |
| Protein Name | Mast/stem cell growth factor receptor Kit |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,134
- Clinical molecules 305
- Avg pChEMBL 7.36
KEGG Pathways (11)
Associated Diseases (7)
Active Molecules (1,134)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VUJQGYIVERKNSC
|
7.9 | IC50 | 2 | — | |
AWROSJBGNHPYIE
|
7.9 | IC50 | 2 | — | |
DZGGGZSDTNTLQN
|
7.9 | IC50 | 5 | Yes | |
ISGHDAOLUCVKHI
|
7.9 | IC50 | 2 | — | |
KOTIZNKRVDGKNU
|
7.9 | IC50 | 2 | Yes | |
OGFUMLMDBRBYKQ
|
7.9 | Ki | 3 | — | |
PHACWCVXLRRZGX
|
7.9 | IC50 | 2 | — | |
RAHBGWKEPAQNFF
|
7.9 | Kd | 26 | — | |
RUAMUEWFVAEXLC
|
7.9 | Ki | 3 | — | |
WOINYYVWAXSXMQ
|
7.9 | IC50 | 4 | Yes | |
LVMAULGVWBINFP
|
7.9 | IC50 | 6 | — | |
XWAAKVKNHUQQFW
|
7.9 | IC50 | 3 | Yes | |
XZXHXSATPCNXJR
|
7.9 | Kd | 165 | Yes | |
KSKHYUVIRUJNSQ
|
7.8 | IC50 | 3 | — | |
MDBBPOZQZACUGK
|
7.8 | IC50 | 6 | Yes | |
MOEODMGOTIIAHE
|
7.8 | IC50 | 5 | — | |
MPVGZUGXCQEXTM
|
7.8 | Kd | 61 | Yes | |
NKKNQMFHKZEGQU
|
7.8 | IC50 | 5 | — | |
SECLOTHQGDJSCB
|
7.8 | IC50 | 5 | Yes | |
UTEPROJRMFGHNF
|
7.8 | Ki | 3 | — | |
XLXUBQMGJVAQIF
|
7.8 | IC50 | 2 | — | |
ZTLCFWVRTDYRQG
|
7.8 | IC50 | 2 | — | |
RAOCKIXJWYDYCO
|
7.8 | IC50 | 5 | Yes | |
DMTDZFGYURLLKX
|
7.8 | IC50 | 13 | Yes | |
DUHSHOMFAWSMPC
|
7.8 | IC50 | 4 | — | |
GXAIYZPLZBVGNJ
|
7.8 | Ki | 3 | — | |
KOSUFZUQHXDTAI
|
7.8 | IC50 | 5 | — | |
MJIIYXFGPPGPGB
|
7.8 | IC50 | 5 | — | |
ZPSQSBRNPLBDHP
|
7.8 | IC50 | 3 | Yes | |
BCDAHFZFGKOCPG
|
7.8 | IC50 | 4 | — | |
FDVSOQRNTAPCHB
|
7.8 | Ki | 40 | — | |
LGHBDVLAHHANMX
|
7.8 | Ki | 53 | — | |
NCJGUXSHLPYQDR
|
7.8 | IC50 | 2 | Yes | |
NODCQQSEMCESEC
|
7.8 | IC50 | 2 | — | |
SHKVYTQIJOOEMA
|
7.8 | IC50 | 6 | — | |
SZPKERXOPUWUPW
|
7.8 | IC50 | 3 | — | |
VCRKDNXOGDJUAN
|
7.8 | IC50 | 4 | Yes | |
VSCYVMFGKQHZQG
|
7.8 | Ki | 3 | — | |
WOKGDWSLHLGJCZ
|
7.8 | IC50 | 3 | Yes | |
XMUWGNAFKPBEAU
|
7.8 | IC50 | 5 | Yes | |
PBQIIKOVMRFZEQ
|
7.8 | IC50 | 3 | Yes | |
PFQKMGZTPAMJKD
|
7.8 | IC50 | 2 | — | |
WTWMNNKZEVJCBK
|
7.8 | IC50 | 5 | — | |
ZMQAYSHYLVAIDP
|
7.8 | IC50 | 2 | — | |
GBJVVSCPOBPEIT
|
7.8 | Kd | 13 | Yes | |
GDCAJIUCFRKHLA
|
7.8 | IC50 | 2 | — | |
MHVFDATVTOZXQW
|
7.8 | IC50 | 6 | Yes | |
NXEKPYWQVKXSPV
|
7.8 | IC50 | 2 | Yes | |
QYZOGCMHVIGURT
|
7.8 | Kd | 26 | Yes | |
SPMHGQZFMNZCBV
|
7.8 | IC50 | 30 | Yes |