Target Details
| UniProt AC | P10721 |
|---|---|
| Gene Symbol | KIT |
| Protein Name | Mast/stem cell growth factor receptor Kit |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,134
- Clinical molecules 305
- Avg pChEMBL 7.36
KEGG Pathways (11)
Associated Diseases (7)
Active Molecules (1,134)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QJIVDCJIPGAKQZ
|
8.0 | Ki | 25 | — | |
RITAVMQDGBJQJZ
|
8.0 | Ki | 33 | — | |
SILANKVZJSUJHJ
|
8.0 | IC50 | 9 | — | |
VBBRNWQCPHQDID
|
8.0 | Ki | 3 | Yes | |
XLYVQVWMTOLDNL
|
8.0 | IC50 | 21 | — | |
XLYVQVWMTOLDNL
|
8.0 | IC50 | 21 | — | |
XOOAAYRIVATZNM
|
8.0 | Ki | 55 | — | |
XPLJEFSRINKZLC
|
8.0 | IC50 | 5 | Yes | |
YESKHRZGFKDGEH
|
8.0 | IC50 | 3 | — | |
YXTDYCAIPCZQMK
|
8.0 | Ki | 3 | — | |
JEGKVDSRNBUXAN
|
8.0 | IC50 | 3 | — | |
FJYFVYKYNSQZCC
|
8.0 | IC50 | 2 | Yes | |
FKFACVZGGDYEHZ
|
8.0 | IC50 | 5 | Yes | |
GWVUCXTYNJIWGK
|
8.0 | Kd | 3 | — | |
INWRCUFOGIVMJS
|
8.0 | Ki | 3 | — | |
MPDAYIPCEWJKOY
|
8.0 | IC50 | 4 | — | |
PUIMLXYJXGFFNV
|
8.0 | IC50 | 4 | — | |
QONPPIZSNSSCSK
|
8.0 | IC50 | 45 | Yes | |
UOEZVMBYMMMIIY
|
8.0 | IC50 | 3 | — | |
UTRWIKREJCMOST
|
8.0 | IC50 | 2 | — | |
XHCPCYVQXFHJAU
|
8.0 | IC50 | 12 | — | |
ZTVQNBOBFFHIID
|
8.0 | Ki | 3 | — | |
PJGPXHUOFQXHSM
|
8.0 | IC50 | 3 | — | |
SPMVMDHWKHCIDT
|
8.0 | IC50 | 30 | — | |
VKBFHTIUXUCYRQ
|
8.0 | Ki | 66 | — | |
RGUQJUZAJQPBOS
|
7.9 | IC50 | 3 | — | |
UWHYTXRXDYNHKS
|
7.9 | Ki | 3 | — | |
GUBJNPWVIUFSTR
|
7.9 | Kd | 103 | — | |
ABBVAIMDGQMDHS
|
7.9 | Ki | 4 | Yes | |
BAFNQSRMVYVKQR
|
7.9 | IC50 | 2 | Yes | |
DIMLYBUSJYNUFT
|
7.9 | IC50 | 6 | — | |
FELCCLMGXTVEGI
|
7.9 | Ki | 4 | Yes | |
JSAIPLUIDULEAD
|
7.9 | Ki | 3 | — | |
LHWABYLWRJNIIY
|
7.9 | IC50 | 7 | — | |
MDHJZTYSOIXDLA
|
7.9 | IC50 | 4 | Yes | |
MEQSMKIFBMBPQX
|
7.9 | IC50 | 6 | Yes | |
MFXYPZFQMDMZNN
|
7.9 | IC50 | 2 | — | |
MIDUFBKQPOWGMC
|
7.9 | IC50 | 5 | Yes | |
PQJDGKYKJGBRBM
|
7.9 | Ki | 5 | Yes | |
UVNBMNWTGOQKQF
|
7.9 | IC50 | 8 | Yes | |
UXYIPHKBTFKDMP
|
7.9 | IC50 | 3 | — | |
XQUGABIPVADSEL
|
7.9 | IC50 | 2 | Yes | |
ZLIFFWATVLSAPF
|
7.9 | IC50 | 2 | — | |
ZUURGOPVVCUCTB
|
7.9 | IC50 | 2 | Yes | |
IJFFMXZETMQIDH
|
7.9 | Ki | 3 | — | |
OJOMKFBUCUYZRW
|
7.9 | IC50 | 3 | — | |
OZSJPXRPIQKJRS
|
7.9 | IC50 | 2 | — | |
WJAXVXBCECPBCW
|
7.9 | IC50 | 3 | — | |
XJNQIRXYMVFKTA
|
7.9 | Ki | 3 | — | |
BRTHUECZMVKNMQ
|
7.9 | IC50 | 7 | — |