Target Details
| UniProt AC | P10721 |
|---|---|
| Gene Symbol | KIT |
| Protein Name | Mast/stem cell growth factor receptor Kit |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,134
- Clinical molecules 305
- Avg pChEMBL 7.36
KEGG Pathways (11)
Associated Diseases (7)
Active Molecules (1,134)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JXXVUIBYJYNDBA
|
8.1 | IC50 | 3 | — | |
LDRYCDRIKRFDRD
|
8.1 | IC50 | 5 | Yes | |
QCUODDVWGHBDKJ
|
8.1 | Ki | 3 | — | |
QXLGSVJYRNECIT
|
8.1 | IC50 | 3 | — | |
QXUCXWRNTARBGK
|
8.1 | IC50 | 3 | — | |
FYTNSFVHUFSPDY
|
8.1 | Ki | 3 | — | |
OEUMLQMTMOCCGW
|
8.1 | Kd | 6 | — | |
PIQCTGMSNWUMAF
|
8.1 | Kd | 137 | Yes | |
ADGOPPKEIZXKAZ
|
8.1 | Ki | 3 | — | |
HDZYCUZNQKCOGY
|
8.1 | IC50 | 3 | — | |
MRAGPKBXJJGPCW
|
8.1 | Ki | 3 | — | |
XGRIDNQIXZILPG
|
8.1 | IC50 | 3 | — | |
MBUPGYAZYBFASN
|
8.1 | IC50 | 2 | Yes | |
MCTXSDCWFQAGFS
|
8.1 | IC50 | 3 | — | |
MHCPAORAYMTGCZ
|
8.1 | Ki | 37 | — | |
RBXYGQNZRVPDNB
|
8.1 | Ki | 34 | — | |
WJEOLQLKVOPQFV
|
8.1 | Kd | 24 | — | |
XKZINYYXWJEYEL
|
8.1 | Ki | 37 | — | |
MJSHVHLADKXCML
|
8.1 | IC50 | 11 | — | |
YMHOIAKNPORUIV
|
8.1 | IC50 | 3 | — | |
HKIJOVMUJUDWGI
|
8.1 | IC50 | 4 | — | |
RHWUJWQTWHXYPV
|
8.1 | IC50 | 3 | — | |
XQKRNUCXAFMEFO
|
8.1 | Ki | 3 | — | |
VWWPJZRYGAVMKS
|
8.1 | IC50 | 3 | — | |
YTHUQGIGAIZNIM
|
8.1 | IC50 | 3 | — | |
KFDIBWHWNIGQSX
|
8.1 | IC50 | 2 | — | |
BMWHAGVKNLRXNW
|
8.1 | IC50 | 3 | — | |
DACQLXDKBYZOIO
|
8.1 | Ki | 3 | — | |
HZIZEKOMOILAJT
|
8.1 | IC50 | 6 | Yes | |
IHZBPVIBWDITMK
|
8.1 | IC50 | 2 | Yes | |
NZUICIGFUCOURS
|
8.1 | IC50 | 4 | — | |
QNSYKQNSCIEOLI
|
8.1 | IC50 | 5 | Yes | |
SHTNULLAAVPXRC
|
8.1 | IC50 | 4 | — | |
UKICZFWMZQMZGK
|
8.1 | IC50 | 3 | Yes | |
VSNJCPXJAHKLRS
|
8.1 | Ki | 7 | Yes | |
WINHZLLDWRZWRT
|
8.1 | Kd | 201 | Yes | |
ZGRFFKUUDPFJDU
|
8.1 | IC50 | 2 | — | |
NJLUOCLXYPXAHG
|
8.0 | Ki | 3 | — | |
SEXVGHCKBMFFSZ
|
8.0 | IC50 | 3 | — | |
MVAYPHGEGDDSJN
|
8.0 | IC50 | 6 | — | |
WRMITRKGBHCESG
|
8.0 | IC50 | 2 | — | |
NEQZWEXWOFPKOT
|
8.0 | IC50 | 9 | Yes | |
JHKCROCKUJZVRL
|
8.0 | IC50 | 2 | — | |
PKDOQGUKLRAMEF
|
8.0 | Ki | 3 | — | |
FGFZBTQWDLZHSI
|
8.0 | IC50 | 4 | — | |
FPQYONGXMYWJCL
|
8.0 | IC50 | 2 | — | |
HQPNLIKXAPLWBQ
|
8.0 | IC50 | 12 | Yes | |
KENMZDPHYLZVEW
|
8.0 | IC50 | 5 | Yes | |
LODWOBAYUQRWKD
|
8.0 | IC50 | 7 | — | |
NMGSBNKYPAIWOG
|
8.0 | IC50 | 3 | — |