Target Details
| UniProt AC | P10721 |
|---|---|
| Gene Symbol | KIT |
| Protein Name | Mast/stem cell growth factor receptor Kit |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,134
- Clinical molecules 305
- Avg pChEMBL 7.36
KEGG Pathways (11)
Associated Diseases (7)
Active Molecules (1,134)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YVRJNNUMUYEWAJ
|
8.3 | IC50 | 2 | — | |
YWSJCLQQBSHJBQ
|
8.3 | IC50 | 2 | — | |
ZGLBORDNOBELSS
|
8.3 | IC50 | 2 | — | |
YOHLRCOPRAVUCJ
|
8.2 | IC50 | 6 | — | |
BVQJGEBCGLWTNC
|
8.2 | Ki | 3 | — | |
MWDKQVZICDCEDA
|
8.2 | IC50 | 3 | — | |
NUAJOPNJJAYNJG
|
8.2 | IC50 | 3 | — | |
OBLBAQUXHOPUQG
|
8.2 | Ki | 3 | — | |
OLGFKJJJBLWTNP
|
8.2 | IC50 | 4 | Yes | |
OWSMSMNEFKFQBZ
|
8.2 | IC50 | 3 | — | |
UUUZEMLVABCSCR
|
8.2 | Ki | 3 | — | |
VZSOVTDSOYVYSF
|
8.2 | IC50 | 3 | — | |
FQEYESALQSIRAQ
|
8.2 | Ki | 3 | — | |
RUPINSRFDWKDBS
|
8.2 | IC50 | 3 | — | |
SDYGMEWQBSWSIW
|
8.2 | IC50 | 6 | — | |
AKRIJSSBKYPXID
|
8.2 | Ki | 3 | — | |
AMHUBFWCCMLLCJ
|
8.2 | IC50 | 15 | — | |
CGWDFIYFJPIFIK
|
8.2 | IC50 | 3 | — | |
DZSUJUOJJJCWGG
|
8.2 | IC50 | 55 | Yes | |
FIJWNTPHEHDJQG
|
8.2 | IC50 | 6 | Yes | |
FQYLJBVSYHZWLT
|
8.2 | IC50 | 35 | Yes | |
IUQURQCHOSRPJM
|
8.2 | IC50 | 4 | Yes | |
NHHQJBCNYHBUSI
|
8.2 | Kd | 220 | — | |
SNGNZNPCCSZZBJ
|
8.2 | IC50 | 3 | Yes | |
WLAVZAAODLTUSW
|
8.2 | IC50 | 7 | — | |
XBBZAHDOGBGKGM
|
8.2 | IC50 | 5 | Yes | |
CAMZXNIVTYLQCA
|
8.2 | Ki | 3 | — | |
LHLGUOHREUTYTO
|
8.2 | IC50 | 4 | Yes | |
NXWOTWQLSTXDFR
|
8.2 | IC50 | 2 | — | |
JPTMGCYMHIJHRQ
|
8.2 | IC50 | 2 | — | |
PHXJVRSECIGDHY
|
8.2 | IC50 | 59 | — | |
CARLZFLTQJQGIP
|
8.2 | IC50 | 3 | — | |
CXQHYVUVSFXTMY
|
8.2 | IC50 | 154 | — | |
KIRQYDLDUZGZPQ
|
8.2 | Ki | 3 | — | |
LKPYVIHIXNNVJX
|
8.2 | IC50 | 3 | — | |
QGLVSYZUEILELT
|
8.2 | IC50 | 3 | — | |
QMCPPBRAJKQPLH
|
8.2 | Ki | 3 | — | |
WQIKRJDLIIEKAG
|
8.2 | IC50 | 2 | — | |
ZNFMAXYFBGIDKY
|
8.2 | IC50 | 3 | — | |
ACBAZTUYTSKGTP
|
8.2 | IC50 | 2 | Yes | |
DGLXOJMLPNCUDE
|
8.2 | IC50 | 7 | Yes | |
GEGCXGMFUYJULA
|
8.2 | IC50 | 30 | Yes | |
LYHXSDWIWVVZPB
|
8.2 | IC50 | 6 | Yes | |
MAXWPKHIRAUGLM
|
8.2 | IC50 | 3 | — | |
QAOMWMNQOYMGAR
|
8.2 | IC50 | 2 | — | |
QKPLUKMJEKRAJD
|
8.2 | IC50 | 30 | Yes | |
SXSIVJXOXSHKPK
|
8.2 | IC50 | 5 | Yes | |
ZJRFZMRNTYZEFF
|
8.2 | IC50 | 2 | — | |
AGENIADQYCDWLP
|
8.1 | Ki | 3 | — | |
HURVYTRTFBZJAW
|
8.1 | IC50 | 2 | — |