Target Details
| UniProt AC | P10721 |
|---|---|
| Gene Symbol | KIT |
| Protein Name | Mast/stem cell growth factor receptor Kit |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,134
- Clinical molecules 305
- Avg pChEMBL 7.36
KEGG Pathways (11)
Associated Diseases (7)
Active Molecules (1,134)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JVSPTGDDSIVSOE
|
8.4 | Ki | 3 | — | |
NFCXPDAZPBFBRT
|
8.4 | Ki | 3 | — | |
OYUDNKFIGXAIRZ
|
8.4 | IC50 | 16 | Yes | |
UZISGDYRMAXEPZ
|
8.4 | IC50 | 5 | — | |
VIHCLUIQGPQVJO
|
8.4 | IC50 | 3 | — | |
WCSWTYSYHRBWDT
|
8.4 | IC50 | 3 | Yes | |
XDDLRMCIDZLHNL
|
8.4 | IC50 | 3 | — | |
QQGKEHCROAPVMW
|
8.4 | IC50 | 3 | — | |
SANPFBFWRPCKIY
|
8.4 | IC50 | 3 | — | |
JYBQEMYHVMILOJ
|
8.4 | IC50 | 5 | — | |
QCKKTDVCCCBGDD
|
8.4 | IC50 | 8 | — | |
RQMAVXSBMSSQDJ
|
8.4 | Ki | 3 | — | |
UGEJLCNSVIVALC
|
8.4 | IC50 | 41 | — | |
FVPYEAORCOKOLV
|
8.4 | IC50 | 6 | — | |
AAUCXXCMBFZYRT
|
8.3 | Kd | 2 | — | |
KRCPKGPVOUOHOW
|
8.3 | IC50 | 3 | — | |
VOEBMPAZQQYYGC
|
8.3 | IC50 | 5 | Yes | |
ONIQOQHATWINJY
|
8.3 | IC50 | 25 | — | |
CAAAKLVRRGRQHX
|
8.3 | Ki | 3 | — | |
PSBGROLQRNSAMY
|
8.3 | IC50 | 2 | — | |
SIXVDPYFTBZLMQ
|
8.3 | IC50 | 2 | — | |
APMQKHHNTLVDQD
|
8.3 | IC50 | 6 | Yes | |
CVWXJKQAOSCOAB
|
8.3 | Kd | 35 | — | |
DEPRXLRJLFPMSV
|
8.3 | IC50 | 2 | — | |
DLYHIJZSZUMFEL
|
8.3 | IC50 | 5 | Yes | |
KGSRYTUWXUESJK
|
8.3 | IC50 | 7 | — | |
KNARVZUUCLIBGV
|
8.3 | Ki | 33 | — | |
MZPQDMUNWXBKLC
|
8.3 | IC50 | 3 | — | |
NSKBZEAMNHXVRQ
|
8.3 | IC50 | 4 | Yes | |
OSMXTIVEGNMCKM
|
8.3 | IC50 | 4 | — | |
OYNIXDXAPYDRHC
|
8.3 | IC50 | 2 | Yes | |
VBXKSTHBDBMAQV
|
8.3 | IC50 | 2 | Yes | |
XBYVOPRDASFDMY
|
8.3 | Ki | 42 | — | |
XEEJFCRYWIMJSK
|
8.3 | IC50 | 2 | — | |
ZGDSBEUMPIMXBM
|
8.3 | Ki | 42 | — | |
BFAFTEXTXVWPSX
|
8.3 | IC50 | 5 | Yes | |
HXPKYBPDEWUZKU
|
8.3 | IC50 | 3 | — | |
HBWUNGZZOZIRLQ
|
8.3 | IC50 | 2 | — | |
AQAZMVVLAOLUPL
|
8.3 | IC50 | 2 | — | |
BHJMKBAJRGNMGC
|
8.3 | IC50 | 2 | — | |
CDDZQGUAUSHZFZ
|
8.3 | IC50 | 2 | — | |
FKNPENIHAAPMRC
|
8.3 | IC50 | 2 | — | |
GMUXDKZNMOZDKO
|
8.3 | IC50 | 2 | — | |
HTIOELJVBGXYQR
|
8.3 | IC50 | 2 | — | |
IQQVFGJWEJAHBR
|
8.3 | IC50 | 2 | — | |
KLOPQHWNVNJIMS
|
8.3 | IC50 | 2 | — | |
MKFKYKXIANOUHV
|
8.3 | IC50 | 2 | — | |
MPDVLCDGYNYLDZ
|
8.3 | IC50 | 2 | — | |
TXNMFHSHEJRKSX
|
8.3 | IC50 | 2 | — | |
XBCQOKINRQAZKD
|
8.3 | IC50 | 2 | — |