Target Details
| UniProt AC | P10721 |
|---|---|
| Gene Symbol | KIT |
| Protein Name | Mast/stem cell growth factor receptor Kit |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00047 (ig) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,134
- Clinical molecules 305
- Avg pChEMBL 7.36
KEGG Pathways (11)
Associated Diseases (7)
Active Molecules (1,134)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MWXLURJNASFGGM
|
8.7 | IC50 | 5 | — | |
OIANGKGOYKDGQV
|
8.7 | Kd | 10 | — | |
KEDANNMRCOENMZ
|
8.6 | IC50 | 7 | — | |
NXQOLSZAEQSUKO
|
8.6 | IC50 | 3 | — | |
PIBOHFLFTZMJME
|
8.6 | IC50 | 2 | — | |
WAKUIUNRDNSMQR
|
8.6 | Kd | 4 | — | |
QODZCSPDZVDCSD
|
8.6 | IC50 | 7 | — | |
RKLGMDOZEOTQEM
|
8.6 | Ki | 12 | — | |
BCABRBNGPCXUDA
|
8.6 | IC50 | 2 | — | |
NLZDIXVVUFRBAV
|
8.6 | IC50 | 2 | — | |
XNFNECKXICLHAD
|
8.6 | IC50 | 2 | — | |
WIVSUJLYDAGUDC
|
8.6 | IC50 | 2 | — | |
ZBNZXTGUTAYRHI
|
8.6 | IC50 | 102 | Yes | |
PETGNDYNMCNUKJ
|
8.6 | IC50 | 3 | — | |
VTWWRKFUHCSCEW
|
8.5 | Kd | 19 | — | |
INOASWZOZPQAQM
|
8.5 | IC50 | 5 | — | |
SEJGTFPOEJWEGG
|
8.5 | Kd | 149 | — | |
CXDOYTGMCAHUID
|
8.5 | IC50 | 2 | Yes | |
FEGRQUWSKADGSP
|
8.5 | IC50 | 6 | Yes | |
FLJOFQUXYAWOPE
|
8.5 | IC50 | 2 | — | |
FLOSOQYXYAJVAG
|
8.5 | IC50 | 2 | — | |
LRUKBEHTGXFIJS
|
8.5 | IC50 | 2 | Yes | |
QJOMTUGNMKUBCP
|
8.5 | IC50 | 3 | — | |
QXMRDWNIKLPTAU
|
8.5 | IC50 | 2 | Yes | |
VCLVPTJGTKXMSP
|
8.5 | IC50 | 2 | — | |
WSBZFFNSBMBYQA
|
8.5 | IC50 | 9 | — | |
VMAAFUOXTWPYRN
|
8.5 | IC50 | 9 | Yes | |
HKZKELVPGXJIMW
|
8.5 | Ki | 41 | — | |
ULHGAQSVFPOUDY
|
8.5 | Ki | 43 | — | |
RITAVMQDGBJQJZ
|
8.5 | Kd | 43 | — | |
SHPFDGWALWEPGS
|
8.5 | Kd | 35 | — | |
GJYUDCNOWIRHBL
|
8.5 | IC50 | 5 | Yes | |
WDAHGVLBPINGHW
|
8.5 | IC50 | 6 | — | |
DXPSQKSTVIVZLV
|
8.5 | IC50 | 6 | Yes | |
LDFNWQUVEYWFOH
|
8.5 | IC50 | 3 | — | |
WNODSYGAOAIJFH
|
8.5 | IC50 | 2 | — | |
JWIPHVWAOYTCOQ
|
8.4 | IC50 | 2 | — | |
NEXXSLYFHONHLW
|
8.4 | IC50 | 2 | — | |
PDSSQGHYCJMBBM
|
8.4 | IC50 | 2 | — | |
BEIAIBOGYLFZCK
|
8.4 | IC50 | 4 | — | |
FDCKDXZISZRERO
|
8.4 | IC50 | 5 | — | |
MDFHFYALOAZVKP
|
8.4 | IC50 | 2 | — | |
BPGIPYJOESFNQI
|
8.4 | IC50 | 6 | Yes | |
CCIRQCXOVCNPBI
|
8.4 | IC50 | 3 | — | |
COXZTUCUTWYLEP
|
8.4 | IC50 | 2 | Yes | |
DIWNHTDZEZGKJK
|
8.4 | IC50 | 3 | — | |
GRDPLDYSIKQSRC
|
8.4 | IC50 | 3 | — | |
GUKDQMJDSRANAC
|
8.4 | IC50 | 2 | — | |
IDFVXZZDQOMMGE
|
8.4 | IC50 | 2 | Yes | |
JBBBYMPMAJVCSI
|
8.4 | IC50 | 3 | Yes |