Target Details
| UniProt AC | P10636 |
|---|---|
| Gene Symbol | MAPT |
| Protein Name | Microtubule-associated protein tau |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00418 (Tubulin-binding) |
Summary
- Multi-target molecules 150
- Clinical molecules 0
- Avg pChEMBL 7.12
KEGG Pathways (4)
Associated Diseases (4)
Active Molecules (150)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CPNUDRZQULAFCT
|
6.7 | Ki | 3 | — | |
DJAGWSNSAWJXLX
|
6.7 | IC50 | 2 | — | |
NOZXPLNYHOGSHE
|
6.6 | Ki | 3 | — | |
UJXWJWJKWZNYSW
|
6.6 | IC50 | 2 | — | |
FGYNZFHVGOFCMD
|
6.6 | IC50 | 2 | — | |
KMXBENJAVFIELJ
|
6.6 | IC50 | 3 | — | |
MNIRHKZCFQNAGM
|
6.6 | IC50 | 3 | — | |
PKBMKQHUGHPUML
|
6.6 | IC50 | 2 | — | |
JKVBLFAUDIBMEH
|
6.5 | IC50 | 3 | — | |
PXMDNOCHJZJAFM
|
6.5 | IC50 | 2 | — | |
UQOZNVGULYNSJW
|
6.5 | IC50 | 2 | — | |
BHTCXYKONZVALL
|
6.5 | Ki | 3 | — | |
MAEBGEQKDJPVBH
|
6.5 | IC50 | 2 | — | |
UXFHOMCAQUWAHI
|
6.5 | IC50 | 3 | — | |
NRVJSTPJGPGYAF
|
6.5 | IC50 | 3 | — | |
RQZPNTQBUCGKFA
|
6.5 | IC50 | 2 | — | |
UFOSROJETSAJRO
|
6.5 | IC50 | 2 | — | |
ZKOUORMEQBYWEC
|
6.5 | IC50 | 2 | — | |
NOZXPLNYHOGSHE
|
6.5 | Ki | 3 | — | |
VRQYMKLREADGJR
|
6.4 | IC50 | 2 | — | |
WPZSQSSOBHCYOZ
|
6.4 | Ki | 3 | — | |
RJSPUDYHVAJALL
|
6.4 | IC50 | 2 | — | |
VPGLALPDHBCDQS
|
6.4 | IC50 | 3 | — | |
QVRAESASNNQBSC
|
6.4 | IC50 | 2 | — | |
SIABTKWBOMYBGS
|
6.4 | IC50 | 2 | — | |
UACJAEPUZXTOBN
|
6.3 | Kd | 2 | — | |
AOIUAVCQCDCNFO
|
6.3 | Ki | 3 | — | |
RQFYFNAGNBUGFC
|
6.3 | IC50 | 3 | — | |
XUIWEDDWEZQAGX
|
6.3 | IC50 | 2 | — | |
FOIHPBSHQSHIIT
|
6.3 | IC50 | 2 | — | |
MREAOFDYHRBSRT
|
6.3 | Ki | 3 | — | |
WPZSQSSOBHCYOZ
|
6.3 | Ki | 3 | — | |
IGJFKRWDBQKNRJ
|
6.2 | IC50 | 2 | — | |
LOASYPPGWUXMEB
|
6.2 | IC50 | 2 | — | |
QAOTWNNTGAUPFL
|
6.2 | IC50 | 2 | — | |
AQOPKQZDRIMOPX
|
6.2 | Ki | 3 | — | |
RBTBFTRPCNLSDE
|
6.2 | IC50 | 5 | — | |
SHJYLIJHYBXPEO
|
6.2 | IC50 | 3 | — | |
OSPFSPHQIOAXEW
|
6.2 | Ki | 3 | — | |
UVTJZQHSPPYGDG
|
6.2 | IC50 | 3 | — | |
VELVOYXHSYTAQT
|
6.2 | Ki | 3 | — | |
MNDLUTPGUCHDRU
|
6.2 | IC50 | 2 | — | |
PPISZIMXPLLQGN
|
6.1 | Ki | 3 | — | |
RSKHAKDCRLZRNZ
|
6.1 | Kd | 2 | — | |
WUTXOFQDICTONV
|
6.1 | IC50 | 3 | — | |
UKWZKQJQFGLRFB
|
6.1 | IC50 | 2 | — | |
VMOSNFMFQKNJPH
|
6.1 | IC50 | 3 | — | |
QFDAPLRSMFECOI
|
6.1 | Kd | 2 | — | |
UGFWJLOCVRHXSF
|
6.0 | IC50 | 3 | — | |
KDUHTFCGEYDKBT
|
6.0 | IC50 | 3 | — |