Target Details
| UniProt AC | P10636 |
|---|---|
| Gene Symbol | MAPT |
| Protein Name | Microtubule-associated protein tau |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00418 (Tubulin-binding) |
Summary
- Multi-target molecules 150
- Clinical molecules 0
- Avg pChEMBL 7.12
KEGG Pathways (4)
Associated Diseases (4)
Active Molecules (150)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YYEIHROTXDFNIC
|
7.3 | IC50 | 2 | — | |
MENVSADYTLLXLP
|
7.2 | IC50 | 6 | — | |
LXLVKFBRQINQCN
|
7.2 | IC50 | 3 | — | |
HVZPHINNUZGJAZ
|
7.2 | IC50 | 3 | — | |
SPTOLQPXVZHQQD
|
7.2 | IC50 | 3 | — | |
KZEUBCUXBNEMSQ
|
7.2 | IC50 | 2 | — | |
NGSGOYFKVYMHAD
|
7.2 | IC50 | 2 | — | |
XYTBUOHYMLZOLR
|
7.2 | IC50 | 2 | — | |
AMOBEFCWUAKOSI
|
7.1 | IC50 | 2 | — | |
BHTCXYKONZVALL
|
7.1 | Ki | 3 | — | |
DVUFESKYOOBJLS
|
7.1 | IC50 | 2 | — | |
LAENBVFKZYAQJP
|
7.1 | IC50 | 2 | — | |
AOIUAVCQCDCNFO
|
7.1 | Ki | 3 | — | |
XDFFVEKPUCXBOI
|
7.1 | IC50 | 2 | — | |
XPJQIGWYDMZIOD
|
7.1 | IC50 | 2 | — | |
GSXIRUIKNXNLAP
|
7.1 | IC50 | 3 | — | |
DHUNWVQYYPMPPG
|
7.1 | IC50 | 2 | — | |
MENVSADYTLLXLP
|
7.1 | IC50 | 2 | — | |
ATMYMANOXIJSDR
|
7.0 | IC50 | 2 | — | |
OXEXOPRYGJGEFF
|
7.0 | IC50 | 2 | — | |
KKUQFANVMIQQGN
|
7.0 | IC50 | 2 | — | |
ZOEPKGAWYBURFM
|
7.0 | IC50 | 2 | — | |
NPBXBJGEHIIUSM
|
7.0 | IC50 | 3 | — | |
SHEVKZDATWMHOR
|
7.0 | IC50 | 2 | — | |
RRXNKIRFKWHJJD
|
7.0 | Ki | 2 | — | |
AQOPKQZDRIMOPX
|
6.9 | Ki | 3 | — | |
DHZZLYIYWJJLRB
|
6.9 | IC50 | 3 | — | |
GCQDVAUTFJHBKP
|
6.9 | IC50 | 2 | — | |
JWHJRYPMAPELPT
|
6.9 | IC50 | 2 | — | |
PYDXUBHPYGQXBU
|
6.9 | IC50 | 3 | — | |
SMVQRETZRLOUFQ
|
6.9 | IC50 | 2 | — | |
WWEHEGICBBJKLI
|
6.9 | IC50 | 3 | — | |
JAZBHABYAFZEPR
|
6.9 | IC50 | 2 | — | |
GOMNONYNAWUWRB
|
6.8 | IC50 | 3 | — | |
IQZQCERNFAXKFQ
|
6.8 | IC50 | 3 | — | |
PQUQTSPOFKEROK
|
6.8 | IC50 | 3 | — | |
LWBQXWADRRVTID
|
6.8 | IC50 | 2 | — | |
NMTZYQHZJFNBJB
|
6.8 | IC50 | 2 | — | |
OSPFSPHQIOAXEW
|
6.8 | Ki | 3 | — | |
CHZARGSIIZBMPM
|
6.8 | IC50 | 3 | — | |
DCGYJAQAXSBBMF
|
6.8 | IC50 | 2 | — | |
DDBPEXIOZILUTR
|
6.8 | IC50 | 2 | — | |
NDAFUJBJGDJBNC
|
6.8 | IC50 | 3 | — | |
ZLWLGUFTYZQJRI
|
6.8 | IC50 | 3 | — | |
GKMDVMDXNKYJRV
|
6.8 | IC50 | 2 | — | |
IXZCGAMHPOYBCA
|
6.8 | Ki | 3 | — | |
AWXGVFDBNXCKQV
|
6.8 | IC50 | 2 | — | |
QCOOCCREMZWFAR
|
6.7 | IC50 | 3 | — | |
PVMJVQIVWNDSCP
|
6.7 | IC50 | 2 | — | |
OYNBEDDKSIPEQC
|
6.7 | IC50 | 3 | — |